SCHEMBL7838604

SCHEMBL7838604

COc1ccc2c(OCc3ccc4c(c3)=CC(=O)N=4)ncnc2n1

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.35
PDE5A O76074 1/20 0.33
ENPP1 P22413 1/20 0.33
CYP1A2 P05177 1/20 0.32
KMT2A Q03164 1/20 0.32
LMNA P02545 2/20 0.32
ALDH1A1 P00352 1/20 0.32
MAPT P10636 1/20 0.32
PKM P14618 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32
ADORA2A P29274 1/20 0.32
ADORA1 P30542 1/20 0.32
KDR P35968 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7839823 0.83 EGFR (0.36) EGFRENPP1CYP1A2KMT2ALMNA
SCHEMBL8814662 0.82 EGFR (0.42) EGFRPDE5AKMT2ALMNAALDH1A1
SCHEMBL8816236 0.77 EGFR (0.57) EGFRKMT2AMAPTKDR
SCHEMBL7821637 0.75 PDE5A (0.40) EGFRPDE5ACYP1A2KMT2ALMNA
SCHEMBL7836815 0.74 MAOB (0.43) EGFRPDE5A
SCHEMBL8815271 0.67 F2 (0.36) KMT2AALDH1A1MAPT
SCHEMBL7350494 0.62 ALDH1A1 (0.37) CYP1A2KMT2ALMNAALDH1A1MAPT
SCHEMBL7837582 0.61 EGFR (0.35) EGFRMAPTKDR
SCHEMBL21339635 0.61 EGFR (0.47) EGFRENPP1CYP1A2KMT2ALMNA
SCHEMBL30940152 0.61 EGFR (0.47) EGFRENPP1CYP1A2KMT2AADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0802914-B1 ARYL- AND HETEROARYL- PURINE AND PYRIDOPYRIMIDINE DERIVATIVES PHARMACIA & UPJOHN SPA (IT) 2001-06-06 EP claimed
EP-0802914-A1 ARYL AND HETEROARYL PURINE COMPOUNDS PHARMACIA & UPJOHN S.p.A. (IT) 1997-10-29 EP claimed
WO-1997018212-A1 ARYL AND HETEROARYL PURINE COMPOUNDS PHARMACIA & UPJOHN S.P.A. (IT) 1997-05-22 WO claimed