SCHEMBL7829931

SCHEMBL7829931

NS(=O)(=O)c1ccc(-n2c[c]cn2)cc1

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CA2 P00918 18/20 0.47
CA1 P00915 17/20 0.47
CA5A P35218 4/20 0.47
CA5B Q9Y2D0 4/20 0.47
CA12 O43570 16/20 0.46
CA9 Q16790 16/20 0.46
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45
LMNA P02545 1/20 0.45
PTGS2 P35354 4/20 0.44
SCN2A Q99250 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4881585 0.71 CA12 (0.57) CA2CA1CA5ACA5BCA12
SCHEMBL17358810 0.71 CHRNA7 (0.58) CA2CA1CA5ACA5BCA12
SCHEMBL671068 0.71 NOTUM (0.44) CA2CA1CA12CA9KDM4E
SCHEMBL2903090 0.71 NOTUM (0.48) KDM4EALDH1A1LMNA
SCHEMBL2752440 0.71 NOTUM (0.44) CA2CA1CA5ACA5BKDM4E
SCHEMBL430176 0.70 GAA (0.42) KDM4EPTGS2
SCHEMBL202948 0.68 CA2 (0.81) CA2CA1CA5ACA5BCA12
SCHEMBL7229570 0.68 NOTUM (0.44) CA2CA12CA9KDM4EALDH1A1
SCHEMBL18109146 0.68 LMNA (0.67) CA2CA1CA5ACA5BCA12
SCHEMBL18118202 0.68 NOTUM (0.55) CA2CA1CA5ACA5BCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1131288-A1 PYRROLIDINE DERIVATIVES-CCR-3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2001-09-12 EP disclosed
US-6166015-A Pyrrolidine derivatives-CCR-3 receptor antagonists SYNTEX (U.S.A.) INC. (US) 2000-12-26 US disclosed
WO-2000031032-A1 PYRROLIDINE DERIVATIVES-CCR-3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2000-06-02 WO disclosed