SCHEMBL4881585

SCHEMBL4881585

NS(=O)(=O)c1ccc(-n2cccn2)cc1

nearest known ligand 0.57

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA12 O43570 3/20 0.57
CA1 P00915 3/20 0.57
CA2 P00918 3/20 0.57
CA9 Q16790 3/20 0.57
NOTUM Q6P988 1/20 0.55
KDM4E B2RXH2 1/20 0.54
ALDH1A1 P00352 1/20 0.54
MAPK1 P28482 1/20 0.54
MAPT P10636 5/20 0.54
KMT2A Q03164 4/20 0.54
MEN1 O00255 3/20 0.54
CHRNA7 P36544 1/20 0.52
POLB P06746 1/20 0.51
TP53 P04637 1/20 0.50
PKM P14618 1/20 0.48
CA5A P35218 1/20 0.48
PTGS2 P35354 1/20 0.48
CA5B Q9Y2D0 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Sulfanilamide SCHEMBL28755036 0.88 CA2 (0.50) CA12CA1CA2CA9NOTUM
SCHEMBL295953 0.84 NOTUM (0.61) NOTUMKDM4EALDH1A1MAPK1MAPT
SCHEMBL3112806 0.82 MAPT (0.57) NOTUMKDM4EALDH1A1MAPK1MAPT
SCHEMBL13836239 0.82 KMT2A (0.55) NOTUMKDM4EALDH1A1MAPK1MAPT
SCHEMBL15664506 0.81 LMNA (0.57) CA12CA1CA2CA9MAPT
SCHEMBL4341894 0.80 NOTUM (0.78) NOTUMKDM4EALDH1A1MAPK1MAPT
SCHEMBL13485837 0.78 MAPT (0.60) CA1CA2NOTUMKDM4EALDH1A1
SCHEMBL8203335 0.78 MAPT (0.54) NOTUMKDM4EALDH1A1MAPK1MAPT
SCHEMBL1661109 0.78 MAPT (0.50) NOTUMKDM4EALDH1A1MAPK1MAPT
SCHEMBL18118212 0.77 CHRNA7 (0.68) CA12CA1CA2CA9KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 38 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12103921-B2 Chemical compounds PFIZER INC. (US) 2024-10-01 US disclosed
US-20230382892-A1 Chemical Compounds PFIZER INC. (US) 2023-11-30 US disclosed
US-11718631-B2 Sulphonamides and compositions thereof for treating conditions associated with NLRP activity NOVARTIS AG (CH) 2023-08-08 US disclosed
US-11718631-B2 Sulphonamides and compositions thereof for treating conditions associated with NLRP activity NOVARTIS AG (CH) 2023-08-08 US disclosed
US-11718631-B2 Sulphonamides and compositions thereof for treating conditions associated with NLRP activity NOVARTIS AG (CH) 2023-08-08 US disclosed
US-11702405-B2 Chemical compounds PFIZER INC. (US) 2023-07-18 US disclosed
US-20220402966-A1 BILE ACID DERIVATIVES AS FXR/TGR5 AGONISTS AND METHODS OF USE THEREOF ENANTA PHARM INC (US) 2022-12-22 US disclosed
EP-3445749-B1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS AG (CH) 2022-12-21 EP disclosed
EP-3445749-B1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS AG (CH) 2022-12-21 EP disclosed
US-20220387397-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS AG (CH) 2022-12-08 US disclosed
US-7419962-B2 3,6-bicyclolides ENANTA PHARMACEUTICALS, INC. (US) 2008-09-02 US disclosed
US-20080200527-A1 Cannabinoid Receptor Modulators CAREX SA (FR) 2008-08-21 US disclosed
US-20080027012-A1 BRIDGED CARBAMATE MACROLIDES ENANTA PHARMACEUTICALS, INC. 2008-01-31 US disclosed
US-20080027012-A1 BRIDGED CARBAMATE MACROLIDES ENANTA PHARMACEUTICALS, INC. 2008-01-31 US disclosed
US-7312201-B2 Tetracyclic bicyclolides ENANTA PHARMACEUTICALS, INC. (US) 2007-12-25 US disclosed
US-7312201-B2 Tetracyclic bicyclolides ENANTA PHARMACEUTICALS, INC. (US) 2007-12-25 US disclosed
US-7291602-B2 11,12-lactone bicyclolides ENANTA PHARMACEUTICALS, INC. (US) 2007-11-06 US disclosed
US-7291602-B2 11,12-lactone bicyclolides ENANTA PHARMACEUTICALS, INC. (US) 2007-11-06 US disclosed
EP-0830133-A1 THERAPEUTIC COMPOSITION FOR ARTHRITIS Takeda Chemical Industries, Ltd. (JP) 1998-03-25 EP disclosed
WO-1996033717-A1 THERAPEUTIC COMPOSITION FOR ARTHRITIS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-10-31 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11702405-B2 Chemical compounds HBZ, HBB, HBS1L CA12 4772/4885CA1 4866/4885CA2 3113/4885
US-20230382892-A1 Chemical Compounds HBZ, HBB, HBS1L CA12 4772/4885CA1 4866/4885CA2 3113/4885
US-20220402966-A1 BILE ACID DERIVATIVES AS FXR/TGR5 AGONISTS AND METHODS OF USE THEREOF GPBAR1, NR1H4, SLC10A1 CA12 2446/4885CA1 1773/4885CA2 1361/4885
US-20220387397-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NLRP1, NLRP3, NOD1 CA12 3146/4885CA1 3842/4885CA2 1337/4885
US-20080200527-A1 Cannabinoid Receptor Modulators CNR1, CNR2, HCRTR2 CA12 1909/4885CA1 1542/4885CA2 1744/4885
US-11718631-B2 Sulphonamides and compositions thereof for treating conditions associated with NLRP activity NLRP1, NLRP3, NOD1 CA12 2416/4885CA1 2501/4885CA2 698/4885
US-20080027012-A1 BRIDGED CARBAMATE MACROLIDES HDAC6, SI, HDAC3 CA12 378/4885CA1 2023/4885CA2 363/4885
US-12103921-B2 Chemical compounds HBZ, HBB, HBS1L CA12 4772/4885CA1 4866/4885CA2 3113/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.