SCHEMBL7830469

SCHEMBL7830469

O=C1Cc2cc(Cc3ncnc4ncccc34)ccc2N1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.42
CYP11B1 P15538 1/20 0.42
CYP11B2 P19099 1/20 0.42
MET P08581 1/20 0.41
PDE3B Q13370 1/20 0.40
PDE3A Q14432 1/20 0.40
HTR1A P08908 1/20 0.40
DRD2 P14416 1/20 0.40
ADRA1D P25100 1/20 0.40
HTR2A P28223 1/20 0.40
ADRA1A P35348 1/20 0.40
ADRA1B P35368 1/20 0.40
MAOB P27338 3/20 0.40
GLO1 Q04760 1/20 0.39
GRIA1 P42261 3/20 0.38
SMYD3 Q9H7B4 1/20 0.38
AHR P35869 1/20 0.38
OPRM1 P35372 1/20 0.37
KDR P35968 1/20 0.36
PARP1 P09874 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7829575 0.82 MAOB (0.47) CYP1A2CYP11B1CYP11B2METPDE3B
SCHEMBL7830473 0.81 PTK2 (0.44) CYP1A2CYP11B1CYP11B2GLO1KDR
SCHEMBL7821491 0.81 CYP1A2 (0.40) CYP1A2CYP11B1CYP11B2METPDE3B
Hydrochloric Acid SCHEMBL7833558 0.81 PTK2 (0.43) CYP1A2CYP11B1CYP11B2GLO1KDR
SCHEMBL7822712 0.80 MAOB (0.39) METPDE3BPDE3AHTR1ADRD2
SCHEMBL7833822 0.78 NEK2 (0.44) CYP1A2CYP11B1CYP11B2METPDE3B
SCHEMBL8930219 0.78 SMYD3 (0.41) METPDE3BPDE3AHTR1ADRD2
SCHEMBL7821656 0.76 MPO (0.37) CYP11B1CYP11B2PARP1
SCHEMBL7833358 0.75 EIF2AK2 (0.43) CYP1A2CYP11B1CYP11B2PDE3BPDE3A
SCHEMBL7822353 0.75 BCL6 (0.57) CYP1A2CYP11B1CYP11B2METKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0802914-B1 ARYL- AND HETEROARYL- PURINE AND PYRIDOPYRIMIDINE DERIVATIVES PHARMACIA & UPJOHN SPA (IT) 2001-06-06 EP claimed
EP-0802914-B1 ARYL- AND HETEROARYL- PURINE AND PYRIDOPYRIMIDINE DERIVATIVES PHARMACIA & UPJOHN SPA (IT) 2001-06-06 EP disclosed
US-5965563-A NOVEL PURINE DERIVATIVES SUCH AS N6-(2-OXINDOL-5-YL) ADENINE, METHODS OF SYNTHESIZING THEM; USE AS TYROSINE KINASE INHIBITORS PHARMACIA & UPJOHN S.P.A. (IT) 1999-10-12 US disclosed