SCHEMBL7833822

SCHEMBL7833822

O=C1Cc2cc(Cc3ncnc4nc[nH]c34)ccc2N1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NEK2 P51955 1/20 0.44
MAOB P27338 3/20 0.40
AHR P35869 1/20 0.39
PDE3B Q13370 1/20 0.39
PDE3A Q14432 1/20 0.39
AKT2 P31751 2/20 0.37
PRKACA P17612 1/20 0.37
PRKACG P22612 1/20 0.37
PRKACB P22694 1/20 0.37
SMYD3 Q9H7B4 1/20 0.36
MET P08581 1/20 0.36
GRIA1 P42261 1/20 0.36
CACNG8 Q8WXS5 1/20 0.36
ALDH1A1 P00352 1/20 0.36
BCL6 P41182 1/20 0.35
CDC7 O00311 2/20 0.35
DBF4 Q9UBU7 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7840701 0.82 CDC7 (0.55) NEK2MAOBAHRPDE3BPDE3A
SCHEMBL7830582 0.81 CDC7 (0.56) ALDH1A1CDC7DBF4CYP1A2
SCHEMBL7830469 0.78 CYP1A2 (0.42) MAOBAHRPDE3BPDE3ASMYD3
SCHEMBL8930219 0.77 SMYD3 (0.41) MAOBAHRPDE3BPDE3ASMYD3
SCHEMBL7834634 0.77 AKT2 (0.40) AKT2PRKACAPRKACGPRKACBALDH1A1
SCHEMBL7822681 0.76 NEK2 (0.46) NEK2MAOBAHRPDE3BPDE3A
SCHEMBL7832613 0.74 CDC7 (0.53) NEK2AHRPDE3BPDE3AALDH1A1
SCHEMBL7840018 0.74 SRC (0.44) NEK2MAOBAHRPDE3BPDE3A
SCHEMBL7822712 0.74 MAOB (0.39) MAOBAHRPDE3BPDE3ASMYD3
SCHEMBL27487825 0.71 AKT2 (0.38) AKT2PRKACAPRKACGPRKACBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0802914-B1 ARYL- AND HETEROARYL- PURINE AND PYRIDOPYRIMIDINE DERIVATIVES PHARMACIA & UPJOHN SPA (IT) 2001-06-06 EP claimed
US-5965563-A NOVEL PURINE DERIVATIVES SUCH AS N6-(2-OXINDOL-5-YL) ADENINE, METHODS OF SYNTHESIZING THEM; USE AS TYROSINE KINASE INHIBITORS PHARMACIA & UPJOHN S.P.A. (IT) 1999-10-12 US claimed
CN-1168138-A Aryl and heteroaryl purine compounds PHARMACIA & UPJOHN SPA (IT) 1997-12-17 CN claimed
EP-0802914-B1 ARYL- AND HETEROARYL- PURINE AND PYRIDOPYRIMIDINE DERIVATIVES PHARMACIA & UPJOHN SPA (IT) 2001-06-06 EP disclosed
US-5965563-A NOVEL PURINE DERIVATIVES SUCH AS N6-(2-OXINDOL-5-YL) ADENINE, METHODS OF SYNTHESIZING THEM; USE AS TYROSINE KINASE INHIBITORS PHARMACIA & UPJOHN S.P.A. (IT) 1999-10-12 US disclosed
CN-1168138-A Aryl and heteroaryl purine compounds PHARMACIA & UPJOHN SPA (IT) 1997-12-17 CN disclosed
EP-0802914-A1 ARYL AND HETEROARYL PURINE COMPOUNDS PHARMACIA & UPJOHN S.p.A. (IT) 1997-10-29 EP disclosed
WO-1997018212-A1 ARYL AND HETEROARYL PURINE COMPOUNDS PHARMACIA & UPJOHN S.P.A. (IT) 1997-05-22 WO disclosed