SCHEMBL8930219

SCHEMBL8930219

O=C1Cc2cc(Cc3ncnc4[nH]ccc34)ccc2N1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 2/20 0.41
BRD4 O60885 1/20 0.41
MAP3K11 Q16584 1/20 0.41
MAOB P27338 3/20 0.40
AHR P35869 1/20 0.39
PDE3B Q13370 1/20 0.39
PDE3A Q14432 1/20 0.39
BCL6 P41182 1/20 0.38
CDK2 P24941 2/20 0.37
AKT1 P31749 2/20 0.37
PTK2 Q05397 1/20 0.37
CDK1 P06493 1/20 0.37
KIT P10721 1/20 0.37
KDR P35968 1/20 0.37
HTR1A P08908 1/20 0.36
DRD2 P14416 1/20 0.36
ADRA1D P25100 1/20 0.36
HTR2A P28223 1/20 0.36
ADRA1A P35348 1/20 0.36
ADRA1B P35368 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7830469 0.78 CYP1A2 (0.42) SMYD3MAOBAHRPDE3BPDE3A
SCHEMBL7833822 0.77 NEK2 (0.44) SMYD3MAP3K11MAOBAHRPDE3B
SCHEMBL8928889 0.77 JAK3 (0.42)
SCHEMBL8929171 0.75 BCL6 (0.60) BCL6PTK2
Hydrochloric Acid SCHEMBL8929519 0.74 BCL6 (0.58) BCL6PTK2
SCHEMBL8929278 0.74 TRPA1 (0.56) MAOBKDRMET
SCHEMBL7822712 0.74 MAOB (0.39) SMYD3MAP3K11MAOBAHRPDE3B
SCHEMBL8929550 0.71 CYP17A1 (0.42) MAP3K11KDR
SCHEMBL3574516 0.70 AHR (0.50) SMYD3MAOBAHRPDE3BPDE3A
SCHEMBL8929582 0.70 CDC7 (0.57) PTK2KDRMET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0795556-A1 4-Substituted pyrrolopyrimidine compounds as tyrosin kinase inhibitors PHARMACIA & UPJOHN S.p.A. (IT) 1997-09-17 EP claimed
EP-0795556-A1 4-Substituted pyrrolopyrimidine compounds as tyrosin kinase inhibitors PHARMACIA & UPJOHN S.p.A. (IT) 1997-09-17 EP disclosed