SCHEMBL7830649

SCHEMBL7830649

COc1cccc(O)c1NCc1nc2ccc(-n3ccnc3)cc2[nH]1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 2/20 0.44
MAOB P27338 2/20 0.44
CBFB Q13951 1/20 0.43
FGFR1 P11362 2/20 0.41
FLT1 P17948 1/20 0.41
F9 P00740 2/20 0.40
KLK1 P06870 1/20 0.39
KLK5 Q9Y337 1/20 0.39
CYP11B1 P15538 2/20 0.39
CYP11B2 P19099 2/20 0.39
CSNK1D P48730 3/20 0.37
CSNK1E P49674 3/20 0.37
NCOA3 Q9Y6Q9 1/20 0.36
ADRB2 P07550 1/20 0.36
ADRB1 P08588 1/20 0.36
ADRB3 P13945 1/20 0.36
PDE5A O76074 2/20 0.36
TBXAS1 P24557 2/20 0.36
PDE3B Q13370 2/20 0.36
PDE3A Q14432 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7834220 0.93 MAOA (0.48) MAOAMAOBCBFBFGFR1FLT1
SCHEMBL7830643 0.93 MAOA (0.42) MAOAMAOBCBFBF9CYP11B1
SCHEMBL7832665 0.91 CBFB (0.49) MAOAMAOBCBFBFGFR1FLT1
SCHEMBL7834212 0.86 MAOA (0.45) MAOAMAOBCBFBFGFR1FLT1
SCHEMBL7831676 0.84 CBFB (0.48) MAOAMAOBCBFBFGFR1FLT1
SCHEMBL7832659 0.83 F9 (0.42) MAOAMAOBCBFBFGFR1FLT1
SCHEMBL7837226 0.83 CBFB (0.46) MAOAMAOBCBFBFGFR1FLT1
SCHEMBL7832841 0.82 MAOA (0.44) MAOAMAOBCBFBFGFR1FLT1
SCHEMBL7836269 0.82 MAOA (0.44) MAOAMAOBCBFBFGFR1FLT1
SCHEMBL7822535 0.81 CYP19A1 (0.45) MAOAMAOBFGFR1F9KLK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0894795-B1 Benzimidazole, benzoxazole and benzothiazole derivatives, their preparation and pharmaceutical compositions containing them ADIR (FR) 2001-06-06 EP disclosed
EP-0894795-A1 Benzimidazole, benzoxazole and benzothiazole derivatives, their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1999-02-03 EP disclosed