SCHEMBL7831354

SCHEMBL7831354

CNC(=O)Nc1snc(Sc2ccccc2)c1C(=O)O

nearest known ligand 0.50

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 13/20 0.50
POLB P06746 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
ALDH1A1 P00352 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
RECQL P46063 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.35
MEN1 O00255 1/20 0.34
HPGD P15428 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3076852 0.90 NTRK1 (0.62) NTRK1ALDH1A1MEN1KMT2A
SCHEMBL7834403 0.81 NTRK1 (0.65) NTRK1ALDH1A1L3MBTL1
SCHEMBL7543844 0.72 NTRK1 (0.47) NTRK1POLBSMN1; SMN2
SCHEMBL3094061 0.72 NTRK1 (0.80) NTRK1
SCHEMBL16866541 0.67 ALDH1A1 (0.55) POLBALDH1A1SMN1; SMN2RECQLMEN1
SCHEMBL10481226 0.67 KMT2A (0.65) POLBTDP1ALDH1A1SMN1; SMN2RECQL
SCHEMBL7833961 0.66 NTRK1 (0.48) NTRK1ALDH1A1L3MBTL1
SCHEMBL3087437 0.65 NTRK1 (0.65) NTRK1
SCHEMBL3089722 0.65 NTRK1 (0.67) NTRK1
SCHEMBL3079365 0.63 NTRK1 (0.63) NTRK1ALDH1A1SMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1084114-A1 ISOTHIAZOLE DERIVATIVES USEFUL AS ANTICANCER AGENTS Pfizer Products Inc. (US) 2001-03-21 EP disclosed
WO-1999062890-A1 ISOTHIAZOLE DERIVATIVES USEFUL AS ANTICANCER AGENTS PFIZER PRODUCTS INC. (US) 1999-12-09 WO disclosed