SCHEMBL7834403

SCHEMBL7834403

CNC(=O)Nc1snc(SCc2ccccc2)c1C(=O)O

nearest known ligand 0.65

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 13/20 0.65
PPARG P37231 5/20 0.48
ALDH1A1 P00352 1/20 0.41
CYP2C9 P11712 1/20 0.41
PKM P14618 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3094061 0.91 NTRK1 (0.80) NTRK1PPARG
SCHEMBL7833961 0.84 NTRK1 (0.48) NTRK1PPARGALDH1A1CYP2C9PKM
SCHEMBL7827670 0.83 KDR (0.51) NTRK1PPARGALDH1A1CYP2C9
SCHEMBL7831354 0.81 NTRK1 (0.50) NTRK1ALDH1A1L3MBTL1
SCHEMBL7820566 0.80 NTRK1 (0.49) NTRK1ALDH1A1L3MBTL1
SCHEMBL3096583 0.78 NTRK1 (0.62) NTRK1CYP2C9
SCHEMBL7543844 0.77 NTRK1 (0.47) NTRK1PPARG
SCHEMBL3087313 0.76 NTRK1 (0.59) NTRK1PPARG
SCHEMBL7827451 0.76 NTRK1 (0.62) NTRK1ALDH1A1
SCHEMBL3087133 0.76 NTRK1 (0.59) NTRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1084114-A1 ISOTHIAZOLE DERIVATIVES USEFUL AS ANTICANCER AGENTS Pfizer Products Inc. (US) 2001-03-21 EP disclosed
WO-1999062890-A1 ISOTHIAZOLE DERIVATIVES USEFUL AS ANTICANCER AGENTS PFIZER PRODUCTS INC. (US) 1999-12-09 WO disclosed