SCHEMBL7831979

SCHEMBL7831979

Cc1nc2ccccc2nc1-n1ccnn1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.49
HRH4 Q9H3N8 1/20 0.46
NOTUM Q6P988 6/20 0.44
TSHR P16473 1/20 0.44
SORD Q00796 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.39
PTPN2 P17706 1/20 0.39
PTPN1 P18031 1/20 0.39
NQO2 P16083 2/20 0.38
MAPT P10636 2/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
KEAP1 Q14145 1/20 0.37
CYP19A1 P11511 1/20 0.36
HCRTR1 O43613 1/20 0.36
HCRTR2 O43614 1/20 0.36
GPR3 P46089 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4759243 0.76 ALDH1A1 (0.45) CYP1A2NOTUMPTPN2PTPN1NQO2
SCHEMBL16113419 0.71 NOTUM (0.47) NOTUML3MBTL1MAPTKDM4EKEAP1
SCHEMBL7018102 0.69 BCHE (0.50) TSHRL3MBTL1MAPTKDM4EALDH1A1
SCHEMBL16113420 0.68 NOTUM (0.47) CYP1A2NOTUMKEAP1CYP19A1HCRTR1
SCHEMBL29364974 0.67 MAPT (0.62) CYP1A2HRH4TSHRL3MBTL1PTPN2
SCHEMBL103601 0.67 MAPT (0.62) CYP1A2HRH4TSHRL3MBTL1PTPN2
SCHEMBL241942 0.67 NOTUM (0.50) CYP1A2NOTUMTSHRALDH1A1KEAP1
Quinoline SCHEMBL27588058 0.67 ALDH1A1 (0.55) NOTUMKDM4EALDH1A1KEAP1CYP19A1
SCHEMBL4760703 0.67 NPC1 (0.45) CYP1A2HRH4NOTUMSORDMAPT
SCHEMBL17768591 0.66 NOTUM (0.35) NOTUMMAPTKDM4EALDH1A1HCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0781279-B1 QUINOXALINEDIONE NMDA RECEPTOR ANTAGONISTS PFIZER LTD (GB) 2001-06-13 EP disclosed