SCHEMBL7832141

SCHEMBL7832141

Cc1[nH]c2ccc(O)c(CN(C)C)c2c1C(=O)OCCc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.48
TSHR P16473 3/20 0.46
KMT2A Q03164 6/20 0.44
MEN1 O00255 5/20 0.44
ALDH1A1 P00352 3/20 0.44
LMNA P02545 2/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
GAA P10253 1/20 0.44
MAPT P10636 1/20 0.44
ESR1 P03372 1/20 0.41
ESR2 Q92731 1/20 0.41
ALOX5 P09917 1/20 0.41
MMP1 P03956 1/20 0.40
MMP2 P08253 1/20 0.40
MMP9 P14780 1/20 0.40
MMP12 P39900 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
GRIN2B Q13224 1/20 0.40
RAB9A P51151 4/20 0.40
HTT P42858 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6317736 0.89 NPSR1 (0.49) NPSR1TSHRKMT2AMEN1ALDH1A1
SCHEMBL7837276 0.85 TSHR (0.50) NPSR1TSHRKMT2AMEN1ALDH1A1
SCHEMBL7832805 0.84 TSHR (0.62) NPSR1TSHRKMT2AMEN1ALDH1A1
SCHEMBL7835009 0.81 TSHR (0.47) NPSR1TSHRKMT2AMEN1ALDH1A1
SCHEMBL7832340 0.81 TSHR (0.48) NPSR1TSHRKMT2AMEN1ALDH1A1
SCHEMBL7825727 0.81 TSHR (0.43) NPSR1TSHRKMT2AMEN1ALDH1A1
SCHEMBL7823730 0.80 TSHR (0.43) NPSR1TSHRKMT2AMEN1ALDH1A1
SCHEMBL7834762 0.80 MEN1 (0.44) NPSR1TSHRKMT2AMEN1ALDH1A1
SCHEMBL7837012 0.80 TSHR (0.47) NPSR1TSHRKMT2AMEN1ALDH1A1
SCHEMBL7838453 0.79 ADRB2 (0.49) NPSR1TSHRKMT2AMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1344270-A Functionalized heterocycles as chemokine receptor modulators THOUSAND YEARS MEDICAMENTS INC (US) 2002-04-10 CN disclosed
EP-1144415-A2 FUNCTIONALIZED HETEROCYCLES AS CHEMOKINE RECEPTOR MODULATORS WARNER-LAMBERT COMPANY (US) 2001-10-17 EP disclosed
WO-2000042045-A2 FUNCTIONALIZED HETEROCYCLES AS CHEMOKINE RECEPTOR MODULATORS WARNER-LAMBERT COMPANY (US) 2000-07-20 WO disclosed