SCHEMBL7832318

SCHEMBL7832318

Cc1nc(Nc2ccc(F)c(F)c2)nc(N2CCc3ccc(Cl)cc3C2C)c1C

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AURKA O14965 3/20 0.35
AURKB Q96GD4 3/20 0.35
APP P05067 3/20 0.34
BRD4 O60885 1/20 0.33
AXL P30530 2/20 0.33
ABL1 P00519 2/20 0.32
BCR P11274 2/20 0.32
BTK Q06187 2/20 0.32
FGFR1 P11362 1/20 0.32
ADRA2A P08913 1/20 0.32
ADRA2B P18089 1/20 0.32
ADRA2C P18825 1/20 0.32
TDP1 Q9NUW8 1/20 0.31
TRPA1 O75762 1/20 0.31
JAK2 O60674 2/20 0.31
DRD2 P14416 1/20 0.31
PTK2 Q05397 1/20 0.31
HTR1A P08908 1/20 0.31
DRD3 P35462 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6159247 0.99 AURKA (0.35) AURKAAURKBAPPBRD4AXL
SCHEMBL6158502 0.91 KMT2A (0.37) AURKAAURKBAPPBRD4ADRA2A
SCHEMBL7858511 0.91 AURKA (0.36) AURKAAURKBAPPAXLABL1
Hydrochloric Acid SCHEMBL6160343 0.91 KMT2A (0.36) AURKAAURKBAPPBRD4ADRA2A
Hydrochloric Acid SCHEMBL6158829 0.91 AURKA (0.35) AURKAAURKBAPPAXLABL1
SCHEMBL7822656 0.89 AURKA (0.36) AURKAAURKBAPPABL1BCR
Hydrochloric Acid SCHEMBL7163241 0.88 AURKA (0.36) AURKAAURKBAPPABL1BCR
SCHEMBL7835940 0.88 MEN1 (0.35) AURKAAURKBAPPBRD4ADRA2A
SCHEMBL7823470 0.87 DRD2 (0.35) BRD4ADRA2AADRA2BADRA2CDRD2
Hydrochloric Acid SCHEMBL6159808 0.87 MEN1 (0.34) AURKAAURKBAPPBRD4ADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1131312-A1 NOVEL PYRIMIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF YUHAN CORPORATION, LTD. (KR) 2001-09-12 EP disclosed
WO-2000029403-A1 NOVEL PYRIMIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF YUHAN CORPORATION (KR) 2000-05-25 WO disclosed