SCHEMBL7833147

SCHEMBL7833147

CC(C)(C)[Si](C)(C)OCc1nc2cnccc2[nH]1

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 9/20 0.35
RAB9A P51151 9/20 0.35
SMN1; SMN2 Q16637 8/20 0.35
TP53 P04637 4/20 0.35
TSHR P16473 1/20 0.35
KDM4C Q9H3R0 1/20 0.35
AAK1 Q2M2I8 1/20 0.34
DDAH1 O94760 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPK1 P28482 2/20 0.33
MAPT P10636 1/20 0.33
MEN1 O00255 1/20 0.33
LMNA P02545 1/20 0.33
GAA P10253 1/20 0.33
HTT P42858 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5214411 0.81 NPC1 (0.55) NPC1RAB9ASMN1; SMN2TP53TSHR
SCHEMBL11955037 0.76 KDM4C (0.40) KDM4CAAK1DDAH1GAA
SCHEMBL18995939 0.75 PKM (0.42) SMN1; SMN2KDM4CDDAH1ALDH1A1GAA
SCHEMBL7833353 0.75
SCHEMBL7836911 0.75 NPC1 (0.35) NPC1RAB9ASMN1; SMN2TP53TSHR
SCHEMBL4240656 0.75 KMT2A (0.36) NPC1RAB9ASMN1; SMN2TP53TSHR
SCHEMBL13508627 0.74 KMT2A (0.54) NPC1RAB9ASMN1; SMN2MAPTMEN1
SCHEMBL8536561 0.74 NPC1 (0.32) NPC1RAB9ASMN1; SMN2
SCHEMBL4245924 0.74 SMN1; SMN2 (0.33) NPC1RAB9ASMN1; SMN2TP53TSHR
SCHEMBL10206036 0.74 DDAH1 (0.59) KDM4CDDAH1GAAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0676398-B1 Heterocyclic compounds having anti-diabetic activity, their preparation and their use SANKYO CO (JP) 2001-10-24 EP disclosed
US-6117893-A Heterocyclic compounds having anti-diabetic activity and their use SANKYO COMPANY, LIMITED (JP) 2000-09-12 US disclosed
EP-1022274-A1 Oxazolidinedione and Thiazolidinedione derivatves, their preparation and their use Sankyo Company Limited (JP) 2000-07-26 EP disclosed
US-5977365-A HYPOGLYCEMIC AGENTS SANKYO COMPANY, LIMITED (JP) 1999-11-02 US disclosed
US-5962470-A Heterocyclic compounds having anti-diabetic activity and their use SANKYO COMPANY, LIMITED (JP) 1999-10-05 US disclosed
US-5834501-A TREATING DIABETES OR HYPERLIPEMIA SANKYO COMPANY, LIMITED (JP) 1998-11-10 US disclosed
US-5739345-A HYPOGLYCEMIC AND ANTIDIABETIC AGENTS SANKYO COMPANY, LIMITED (JP) 1998-04-14 US disclosed
US-5624935-A ANTIDIABETIC AGENTS, HYPOGLYCEMIC AGENTS OR ANTILIPEMIC AGENTS SANKYO COMPANY, LIMITED 1997-04-29 US disclosed
EP-0676398-A2 Heterocyclic compounds having anti-diabetic activity, their preparation and their use SANKYO COMPANY LIMITED (JP) 1995-10-11 EP disclosed