SCHEMBL7833583

SCHEMBL7833583

CCOc1ccc([N+](=O)[O-])c(NC)n1

nearest known ligand 0.61

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAOA P21397 4/20 0.61
MAOB P27338 2/20 0.61
LMNA P02545 3/20 0.45
GALR2 O43603 1/20 0.45
POLB P06746 1/20 0.45
TXNRD1 Q16881 6/20 0.43
MAPT P10636 4/20 0.43
ALDH1A1 P00352 3/20 0.43
NPC1 O15118 3/20 0.40
RAB9A P51151 3/20 0.40
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
GSR P00390 1/20 0.39
MAPK1 P28482 2/20 0.38
NFKB1 P19838 1/20 0.38
NFKB2 Q00653 1/20 0.38
RELA Q04206 1/20 0.38
RECQL P46063 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2305462 0.83 MAOA (0.54) MAOAMAOBLMNAGALR2POLB
SCHEMBL2306805 0.83 TXNRD1 (0.54) LMNAGALR2POLBTXNRD1MAPT
SCHEMBL13730216 0.82 MAOA (0.57) MAOAMAOBLMNAPOLBMAPT
SCHEMBL7834233 0.82 MAOA (0.49) MAOAMAOBTXNRD1MAPTNPC1
SCHEMBL7833656 0.80 LMNA (0.46) MAOAMAOBLMNAGALR2POLB
SCHEMBL29535900 0.80 MAOA (0.51) MAOAMAOBPOLBTXNRD1MAPT
SCHEMBL22719062 0.80 MAOA (0.51) MAOAMAOBPOLBTXNRD1MAPT
SCHEMBL11362288 0.80 MAOA (0.51) MAOAMAOBLMNATXNRD1MAPT
SCHEMBL11362292 0.80 MAOA (0.51) MAOAMAOBLMNATXNRD1MAPT
SCHEMBL10743303 0.80 MAOA (0.49) MAOAMAOBLMNATXNRD1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0676398-B1 Heterocyclic compounds having anti-diabetic activity, their preparation and their use SANKYO CO (JP) 2001-10-24 EP disclosed
US-6117893-A Heterocyclic compounds having anti-diabetic activity and their use SANKYO COMPANY, LIMITED (JP) 2000-09-12 US disclosed
EP-1022274-A1 Oxazolidinedione and Thiazolidinedione derivatves, their preparation and their use Sankyo Company Limited (JP) 2000-07-26 EP disclosed
US-5977365-A HYPOGLYCEMIC AGENTS SANKYO COMPANY, LIMITED (JP) 1999-11-02 US disclosed
US-5962470-A Heterocyclic compounds having anti-diabetic activity and their use SANKYO COMPANY, LIMITED (JP) 1999-10-05 US disclosed
US-5834501-A TREATING DIABETES OR HYPERLIPEMIA SANKYO COMPANY, LIMITED (JP) 1998-11-10 US disclosed
US-5739345-A HYPOGLYCEMIC AND ANTIDIABETIC AGENTS SANKYO COMPANY, LIMITED (JP) 1998-04-14 US disclosed
US-5624935-A ANTIDIABETIC AGENTS, HYPOGLYCEMIC AGENTS OR ANTILIPEMIC AGENTS SANKYO COMPANY, LIMITED 1997-04-29 US disclosed
EP-0676398-A2 Heterocyclic compounds having anti-diabetic activity, their preparation and their use SANKYO COMPANY LIMITED (JP) 1995-10-11 EP disclosed
EP-0257399-B1 HAIR DYEING COMPOSITION Beratungslabor für die kosmetische und pharmazeutische Industrie Dipl.-Ing. Karlheinz Schrader (DE) 1991-01-02 EP disclosed
EP-0136730-B1 2-AMINONITROPYRIDINE DERIVATIVES AND PROCESS FOR THE PREPARATION THEREOF RÜTGERSWERKE AKTIENGESELLSCHAFT (DE) 1988-04-27 EP disclosed
EP-0257399-A2 Hair dyeing composition Beratungslabor für die kosmetische und pharmazeutische Industrie Dipl.-Ing. Karlheinz Schrader (DE) 1988-03-02 EP disclosed
EP-0137524-B1 HAIR DYEING COMPOSITIONS RÜTGERSWERKE AKTIENGESELLSCHAFT (DE) 1988-01-20 EP disclosed
US-4567272-A Pyrrole containing 2-aminonitropyridine derivatives RUTGERSWERKE AKTIENGESELLSCHAFT (DE) 1986-01-28 US disclosed
EP-0137524-A1 Hair dyeing compositions RÜTGERSWERKE AKTIENGESELLSCHAFT (DE) 1985-04-17 EP disclosed
EP-0136730-A1 2-Aminonitropyridine derivatives and process for the preparation thereof RÜTGERSWERKE AKTIENGESELLSCHAFT (DE) 1985-04-10 EP disclosed