SCHEMBL7833593

SCHEMBL7833593

CCc1ccc2ccc(CO)cc2n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 1/20 0.45
CYSLTR1 Q9Y271 2/20 0.43
GPBAR1 Q8TDU6 2/20 0.43
CCR1 P32246 1/20 0.36
GAA P10253 1/20 0.36
RPS6KA5 O75582 1/20 0.35
TERT O14746 1/20 0.35
CA12 O43570 1/20 0.35
CA2 P00918 1/20 0.35
CA3 P07451 1/20 0.35
CA4 P22748 1/20 0.35
CA6 P23280 1/20 0.35
CA5A P35218 1/20 0.35
CA7 P43166 1/20 0.35
CA9 Q16790 1/20 0.35
CA14 Q9ULX7 1/20 0.35
CA5B Q9Y2D0 1/20 0.35
PARP1 P09874 1/20 0.35
ELANE P08246 1/20 0.35
CYP1A2 P05177 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9697024 0.87 CYSLTR1 (0.42) HSD17B10CYSLTR1GPBAR1CCR1GAA
SCHEMBL2756576 0.86 CYP1A2 (0.47) HSD17B10GAATERTPARP1ELANE
SCHEMBL16601918 0.77 TERT (0.43) HSD17B10CYSLTR1GPBAR1CCR1GAA
SCHEMBL29970876 0.77 MEN1 (0.46) CYSLTR1GPBAR1GAATERTPARP1
SCHEMBL9458710 0.75 HSD17B10 (0.40) HSD17B10GAARPS6KA5CA12CA2
SCHEMBL13349518 0.75 HSD17B10 (0.44) HSD17B10CYSLTR1GPBAR1CA12CA2
SCHEMBL16284370 0.75 CYP1A2 (0.57) HSD17B10GAATERTELANECYP1A2
SCHEMBL23283355 0.74 NCF1 (0.50) HSD17B10CA12CA2CA3CA4
SCHEMBL12824284 0.73 CYP1A2 (0.50) GAATERTELANECYP1A2CYP2A6
SCHEMBL17179408 0.73 BACE1 (0.52) CYSLTR1GPBAR1TERTPARP1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5444071-A Hypotensive agent IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1995-08-22 US claimed
EP-0412848-B1 Quinoline derivatives, process for their preparation and their use as medicaments ICI PLC (GB) 1995-01-18 EP claimed
CN-1050187-A New quinoline compound and preparation method thereof ICI PLC (GB) 1991-03-27 CN claimed
EP-0412848-A2 Quinoline derivatives, process for their preparation and their use as medicaments ZENECA LIMITED (GB) 1991-02-13 EP claimed
EP-0470795-B2 Process for the manufacture of nitriles AVECIA LTD (GB) 2001-02-21 EP disclosed
US-5444071-A Hypotensive agent IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1995-08-22 US disclosed
EP-0470795-B1 Process for the manufacture of nitriles ZENECA LTD (GB) 1995-01-25 EP disclosed
EP-0470794-B1 Process for the preparation of nitriles ZENECA LTD (GB) 1995-01-25 EP disclosed
EP-0412848-B1 Quinoline derivatives, process for their preparation and their use as medicaments ICI PLC (GB) 1995-01-18 EP disclosed
CN-1059516-A The preparation method of biphenylcarbonitriles ICI LTD (GB) 1992-03-18 CN disclosed
CN-1058965-A The method for preparing new quinoline ICI PLC (GB) 1992-02-26 CN disclosed
EP-0470795-A1 Process for the manufacture of nitriles ZENECA LIMITED (GB) 1992-02-12 EP disclosed
EP-0470794-A1 Process for the preparation of nitriles ZENECA LIMITED (GB) 1992-02-12 EP disclosed
CN-1050187-A New quinoline compound and preparation method thereof ICI PLC (GB) 1991-03-27 CN disclosed
EP-0412848-A2 Quinoline derivatives, process for their preparation and their use as medicaments ZENECA LIMITED (GB) 1991-02-13 EP disclosed