SCHEMBL7833798

SCHEMBL7833798

CCOC(=O)CC(NC(=O)CNC(=O)c1cccc(NC(=N)N)c1)c1ccc(C)s1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.43
POLB P06746 1/20 0.43
NPSR1 Q6W5P4 1/20 0.38
ITGB3 P05106 4/20 0.37
ITGB1 P05556 3/20 0.37
ITGAV P06756 3/20 0.37
ITGA5 P08648 3/20 0.37
ITGB5 P18084 2/20 0.37
ITGB6 P18564 2/20 0.37
ITGB8 P26012 2/20 0.37
ITGA8 P53708 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
HPGD P15428 1/20 0.37
KMT2A Q03164 4/20 0.37
MEN1 O00255 3/20 0.37
F2 P00734 1/20 0.37
F7 P08709 1/20 0.37
KDM4E B2RXH2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7823060 0.92 ITGB3 (0.38) ALDH1A1POLBNPSR1ITGB3ITGB1
SCHEMBL6777666 0.90 ITGB3 (0.47) ALDH1A1POLBITGB3ITGB1ITGAV
SCHEMBL3839471 0.88 GPR139 (0.47) ITGB3ITGB1ITGAVITGA5KMT2A
SCHEMBL7340065 0.87 F7 (0.38) ALDH1A1POLBNPSR1ITGB3ITGB1
SCHEMBL7340341 0.85 F7 (0.41) POLBNPSR1ITGB3ITGB1ITGAV
SCHEMBL7341726 0.85 GPR139 (0.42) ALDH1A1NPSR1ITGB3ITGB1ITGAV
SCHEMBL7340506 0.84 ITGB3 (0.49) ALDH1A1POLBNPSR1ITGB3ITGB1
SCHEMBL7337752 0.84 NPC1 (0.44) ALDH1A1POLBNPSR1ITGB3ITGB1
SCHEMBL7344055 0.83 F7 (0.46) ALDH1A1F2F7GPR139F10
SCHEMBL7341087 0.83 GPR139 (0.48) ITGB3ITGB1ITGAVITGA5ITGB5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0850221-B1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS SEARLE & CO (US) 2001-07-18 EP claimed