SCHEMBL7834192

SCHEMBL7834192

CCOC(=O)c1[nH]c2ccc(Cl)cc2c1CC#N

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.60
CYP1A2 P05177 1/20 0.60
HPGD P15428 1/20 0.60
XBP1 P17861 1/20 0.60
CYP2C19 P33261 1/20 0.60
ALOX15 P16050 9/20 0.54
CNR2 P34972 2/20 0.52
TUBB4A P04350 1/20 0.52
TUBB P07437 1/20 0.52
TUBA3C P0DPH7 1/20 0.52
TUBA1B P68363 1/20 0.52
TUBA4A P68366 1/20 0.52
TUBB4B P68371 1/20 0.52
TUBB3 Q13509 1/20 0.52
TUBB2A Q13885 1/20 0.52
TUBB8 Q3ZCM7 1/20 0.52
TUBA3E Q6PEY2 1/20 0.52
TUBA1A Q71U36 1/20 0.52
TUBA1C Q9BQE3 1/20 0.52
TUBB6 Q9BUF5 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15649200 0.87 ALDH1A1 (0.56) ALDH1A1CYP1A2HPGDXBP1CYP2C19
SCHEMBL12496609 0.86 ALDH1A1 (0.66) ALDH1A1CYP1A2HPGDXBP1CYP2C19
SCHEMBL3954004 0.85 ALDH1A1 (0.68) ALDH1A1CYP1A2HPGDTUBB4ATUBB
SCHEMBL4614808 0.84 ALDH1A1 (0.63) ALDH1A1CYP1A2HPGDXBP1CYP2C19
SCHEMBL7838931 0.83 ALOX15 (0.46) ALDH1A1CYP1A2HPGDXBP1CYP2C19
SCHEMBL9189433 0.83 ALDH1A1 (0.65) ALDH1A1CYP1A2HPGDXBP1CYP2C19
SCHEMBL12326581 0.83 HTR6 (0.67) ALDH1A1HPGDTUBB4ATUBBTUBA3C
SCHEMBL15622584 0.82 ALDH1A1 (0.61) ALDH1A1CYP1A2HPGDXBP1CYP2C19
SCHEMBL21264669 0.81 ALDH1A1 (0.66) ALDH1A1CYP1A2HPGDXBP1CYP2C19
SCHEMBL15622511 0.81 ALDH1A1 (0.63) ALDH1A1CYP1A2HPGDXBP1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015044928-A1 SUBSTITUTED INDOLES AND THEIR USE AS NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS STELLENBOSCH UNIVERSITY (ZA) 2015-04-02 WO disclosed
EP-1147110-A1 PYRAZINO(AZA)INDOLE DERIVATIVES VERNALIS RESEARCH LIMITED (GB) 2001-10-24 EP disclosed
WO-2000044753-A1 PIRAZINO(AZA)INDOLE DERIVATIVES VERNALIS RESEARCH LIMITED (GB) 2000-08-03 WO disclosed