SCHEMBL7834394

SCHEMBL7834394

O=C(NO)c1ccc(OCc2nc3ccc(-n4ccnc4)cc3[nH]2)cc1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C19 P33261 1/20 0.50
F9 P00740 6/20 0.46
CBFB Q13951 1/20 0.45
HDAC6 Q9UBN7 3/20 0.43
HDAC1 Q13547 1/20 0.42
PDE10A Q9Y233 1/20 0.42
SIRT2 Q8IXJ6 1/20 0.41
SIRT1 Q96EB6 1/20 0.41
SIRT3 Q9NTG7 1/20 0.41
ADRB2 P07550 1/20 0.41
ADRB1 P08588 1/20 0.41
ADRB3 P13945 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7834392 0.93 ALDH1A1 (0.50) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL7833681 0.89 ADH5 (0.48) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL7830518 0.83 CBFB (0.50) CYP1A2CYP3A4CYP2D6CYP2C19CBFB
SCHEMBL7831108 0.83 SMN1; SMN2 (0.55) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL7834561 0.83 RAB9A (0.56) CYP1A2CYP3A4CYP2D6CYP2C19F9
SCHEMBL7821732 0.83 RAB9A (0.58) ALDH1A1CYP1A2CYP3A4CYP2D6CBFB
SCHEMBL2619416 0.83 PARP1 (0.45) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C19
Hydrochloric Acid SCHEMBL8148415 0.82 CBFB (0.49) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C19
Hydrochloric Acid SCHEMBL8142735 0.82 SMN1; SMN2 (0.54) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C19
Hydrochloric Acid SCHEMBL8149755 0.82 RAB9A (0.55) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0894795-B1 Benzimidazole, benzoxazole and benzothiazole derivatives, their preparation and pharmaceutical compositions containing them ADIR (FR) 2001-06-06 EP disclosed
US-6040327-A INHIBITORS OF INTERLEUKINS; TREATING RHEUMATOID ARTHRITIS OR ARTHROSIS ADIR ET COMPAGNIE (FR) 2000-03-21 US disclosed
EP-0894795-A1 Benzimidazole, benzoxazole and benzothiazole derivatives, their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1999-02-03 EP disclosed