SCHEMBL7834955

SCHEMBL7834955

CSC1(Cc2ccccc2)C(=O)Nc2ccccc21

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.48
LMNA P02545 2/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
PDK2 Q15119 1/20 0.46
PDK4 Q16654 1/20 0.46
ALDH1A1 P00352 2/20 0.43
KDM4E B2RXH2 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
MAPT P10636 1/20 0.43
CYP2C9 P11712 1/20 0.43
HPGD P15428 1/20 0.43
CYP2C19 P33261 1/20 0.43
CACNA1B Q00975 1/20 0.43
APBA1 Q02410 1/20 0.43
POLB P06746 1/20 0.40
PGR P06401 1/20 0.40
HTT P42858 1/20 0.40
CHRM2 P08172 1/20 0.40
ADORA3 P0DMS8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12165522 0.76 ATM (0.77) ATMLMNASMN1; SMN2PDK2PDK4
SCHEMBL7834463 0.76 PGR (0.59) ATMLMNASMN1; SMN2PDK2PDK4
SCHEMBL28010729 0.72 ATM (0.48) ATMLMNASMN1; SMN2PDK2PDK4
SCHEMBL28010767 0.72 ALDH1A1 (0.67) ATMLMNASMN1; SMN2PDK2PDK4
SCHEMBL11430300 0.72 PDK2 (0.59) LMNASMN1; SMN2PDK2PDK4ALDH1A1
SCHEMBL7836579 0.69 PDK2 (0.60) LMNASMN1; SMN2PDK2PDK4ALDH1A1
SCHEMBL11442529 0.68 PDK2 (0.53) ATMLMNASMN1; SMN2PDK2PDK4
SCHEMBL24281081 0.67 SMN1; SMN2 (0.62) ATMLMNASMN1; SMN2PDK2PDK4
SCHEMBL3244982 0.66 ATM (0.58) ATMLMNASMN1; SMN2PDK2PDK4
SCHEMBL7835297 0.66 PDK2 (0.50) LMNASMN1; SMN2PDK2PDK4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0780388-B1 5HT1Dalpha and 5HT2A ligands LILLY CO ELI (GB) 2001-08-16 EP disclosed
US-5773448-A NERVOUS SYSTEM DISORDERS ELI LILLY AND COMPANY LIMITED (GB) 1998-06-30 US disclosed
EP-0780388-A1 5HT1Dalpha and 5HT2A ligands LILLY INDUSTRIES LIMITED (GB) 1997-06-25 EP disclosed