SCHEMBL783496

SCHEMBL783496

O=C(Nc1ccc(Oc2ccnc(NC(=S)N3CCOCC3)c2)c(F)c1)c1ccnn(-c2ccccc2)c1=O

nearest known ligand 0.55

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AXL P30530 9/20 0.55
MET P08581 14/20 0.53
RIPK2 O43353 1/20 0.51
RIPK1 Q13546 1/20 0.51
RIPK3 Q9Y572 1/20 0.51
KDR P35968 2/20 0.50
MERTK Q12866 5/20 0.48
TYRO3 Q06418 4/20 0.47
BRAF P15056 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2680338 0.89 MET (0.65) AXLMETRIPK2RIPK1RIPK3
SCHEMBL199864 0.87 AXL (0.61) AXLMETRIPK2RIPK1RIPK3
SCHEMBL783423 0.81 MET (0.65) AXLMETRIPK2RIPK1RIPK3
SCHEMBL2742632 0.76 MET (0.77) AXLMETKDRMERTKTYRO3
SCHEMBL199488 0.76 MET (0.76) AXLMETKDR
SCHEMBL1471850 0.75 MET (0.59) AXLMETRIPK2RIPK1RIPK3
SCHEMBL783531 0.73 MET (0.71) AXLMETRIPK2RIPK1RIPK3
SCHEMBL13861033 0.73 MET (0.65) AXLMETKDR
SCHEMBL1471740 0.72 AXL (0.56) AXLMETRIPK2RIPK1RIPK3
SCHEMBL199597 0.72 MET (0.69) METKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1881976-B1 SUBSTITUTED AMIDE DERIVATIVES AS PROTEIN KINASE INHIBITORS AMGEN INC (US) 2012-10-17 EP disclosed
US-20120070413-A1 METHOD OF TREATING CANCER WITH SUBSTITUTED AMIDE DERIVATIVES KIM TAE-SEONG (US) 2012-03-22 US disclosed
US-20120070413-A1 METHOD OF TREATING CANCER WITH SUBSTITUTED AMIDE DERIVATIVES KIM TAE-SEONG (US) 2012-03-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120070413-A1 METHOD OF TREATING CANCER WITH SUBSTITUTED AMIDE DERIVATIVES HGF, HGFAC, MET AXL 855/4885MET 3/4885RIPK2 4290/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.