SCHEMBL7835665

SCHEMBL7835665

CCOC(=O)CC(NC(=O)CNC(=O)c1cccc(NC(=N)N)c1)c1cccnc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 5/20 0.45
ITGA2B P08514 4/20 0.45
ROCK2 O75116 1/20 0.43
ALDH1A1 P00352 1/20 0.41
MAPT P10636 1/20 0.41
NPC1 O15118 1/20 0.41
HPGD P15428 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
SUCNR1 Q9BXA5 2/20 0.40
GPR139 Q6DWJ6 1/20 0.39
ITGAV P06756 3/20 0.39
BRAF P15056 1/20 0.39
POLB P06746 1/20 0.38
ITGB1 P05556 1/20 0.38
ITGA5 P08648 1/20 0.38
ITGB5 P18084 1/20 0.38
ITGB6 P18564 1/20 0.38
ITGB8 P26012 1/20 0.38
ITGA8 P53708 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7339949 0.93 ROCK2 (0.44) ITGB3ITGA2BROCK2ALDH1A1MAPT
SCHEMBL6773670 0.92 ROCK2 (0.43) ITGB3ITGA2BROCK2ALDH1A1MAPT
SCHEMBL7832728 0.91 ROCK2 (0.42) ITGB3ITGA2BROCK2ALDH1A1MAPT
SCHEMBL7341019 0.90 ITGB3 (0.46) ITGB3ITGA2BROCK2ALDH1A1MAPT
SCHEMBL3839471 0.90 GPR139 (0.47) ITGB3ITGA2BGPR139ITGAVITGB1
SCHEMBL7832621 0.89 ITGB3 (0.44) ITGB3ITGA2BROCK2ALDH1A1MAPT
SCHEMBL6772228 0.89 GPR139 (0.43) ITGB3ITGA2BROCK2ALDH1A1MAPT
SCHEMBL6776653 0.88 ITGB3 (0.58) ITGB3ITGA2BSUCNR1ITGAVITGB1
SCHEMBL7340347 0.88 ITGB3 (0.41) ITGB3ITGA2BROCK2ALDH1A1HPGD
SCHEMBL7341726 0.87 GPR139 (0.42) ITGB3ALDH1A1GPR139ITGAVITGB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0850221-B1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS SEARLE & CO (US) 2001-07-18 EP claimed
EP-0850221-B1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS SEARLE & CO (US) 2001-07-18 EP disclosed