SCHEMBL7835767

SCHEMBL7835767

CC(NC(=O)c1ccc(C#N)cc1)C(C)(C)C(=O)O

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PRSS1 P07477 5/20 0.56
CTSG P08311 5/20 0.56
CTRB1 P17538 5/20 0.56
CMA1 P23946 5/20 0.56
MEN1 O00255 1/20 0.56
KMT2A Q03164 1/20 0.56
TRPA1 O75762 2/20 0.49
EPHX2 P34913 1/20 0.47
GSK3B P49841 1/20 0.45
S1PR4 O95977 1/20 0.44
S1PR3 Q99500 1/20 0.44
XDH P47989 1/20 0.44
MAP4K4 O95819 1/20 0.44
MINK1 Q8N4C8 1/20 0.44
TNIK Q9UKE5 1/20 0.44
PPARA Q07869 1/20 0.44
ALDH1A1 P00352 1/20 0.43
PKM P14618 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7837407 0.86 PRSS1 (0.54) PRSS1CTSGCTRB1CMA1MEN1
SCHEMBL16234826 0.82 PRSS1 (0.50) PRSS1CTSGCTRB1CMA1MEN1
SCHEMBL7837711 0.82 CTSG (0.57) PRSS1CTSGCTRB1CMA1MEN1
SCHEMBL7825862 0.81 CTSG (0.80) PRSS1CTSGCTRB1CMA1MEN1
SCHEMBL7825623 0.80 CTSG (0.61) PRSS1CTSGCTRB1CMA1MEN1
SCHEMBL7837210 0.80 CTSG (0.60) PRSS1CTSGCTRB1CMA1MEN1
SCHEMBL12468782 0.79 TRPA1 (0.49) PRSS1CTSGCTRB1CMA1MEN1
SCHEMBL12783210 0.79 MEN1 (0.67) PRSS1CTSGCTRB1CMA1MEN1
SCHEMBL7836801 0.78 CTSG (0.64) PRSS1CTSGCTRB1CMA1MEN1
SCHEMBL7835603 0.78 CTSG (0.63) PRSS1CTSGCTRB1CMA1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0800516-B1 FIBRINOGEN RECEPTOR ANTAGONISTS HAVING SUBSTITUTED (b)-AMINO ACID RESIDUES AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME NIPPON STEEL CORP (JP) 2001-09-19 EP disclosed
US-5866592-A Fibrinogen receptor antagonist and pharmaceutical compositions comprising the same NIPPON STEEL CORPORATION (JP) 1999-02-02 US disclosed