SCHEMBL7835841

SCHEMBL7835841

Cc1nccn1Cc1ccc2[nH]cc(C3CNC3)c2c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 3/20 0.58
HTR2C P28335 2/20 0.58
HTR1D P28221 11/20 0.44
HTR1B P28222 11/20 0.44
LMNA P02545 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
OPRM1 P35372 1/20 0.36
OPRK1 P41145 1/20 0.36
OPRL1 P41146 1/20 0.36
GABRP O00591 1/20 0.36
GABRD O14764 1/20 0.36
GABRA1 P14867 1/20 0.36
GABRB1 P18505 1/20 0.36
GABRG2 P18507 1/20 0.36
GABRB3 P28472 1/20 0.36
GABRA5 P31644 1/20 0.36
GABRA3 P34903 1/20 0.36
GABRA2 P47869 1/20 0.36
GABRB2 P47870 1/20 0.36
GABRA4 P48169 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7831800 0.88 HTR1A (0.57) HTR1AHTR2CHTR1DHTR1BLMNA
SCHEMBL27343955 0.86 HTR1A (0.53) HTR1AHTR2CHTR1DHTR1BLMNA
SCHEMBL8784342 0.84 HTR1A (0.53) HTR1AHTR2CHTR1DHTR1BGABRP
SCHEMBL9545340 0.81 HTR1A (0.41) HTR1AHTR2CHTR1DHTR1BOPRK1
SCHEMBL9087213 0.79 HTR1A (0.42) HTR1AHTR2CLMNAL3MBTL1FLT3
SCHEMBL9086672 0.76 HTR1A (0.59) HTR1AHTR2CHTR1DHTR1BLMNA
SCHEMBL8883273 0.75 HTR1A (0.76) HTR1AHTR2CHTR1DHTR1BCYP1A2
SCHEMBL8783856 0.73 HTR1A (1.00) HTR1AHTR2CHTR1DHTR1B
SCHEMBL8783749 0.70 GABRP (0.56) HTR1AHTR2CHTR1DHTR1BGABRP
SCHEMBL7836170 0.69 HTR1A (0.58) HTR1AHTR2CHTR1DHTR1BCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0630374-B1 IMIDAZOLE, TRIAZOLE AND TETRAZOLE DERIVATIVES MERCK SHARP & DOHME (GB) 2001-09-05 EP disclosed