SCHEMBL9545340

SCHEMBL9545340

CC(C)(C)OC(=O)N1CC(CC=O)C1.Cc1nccn1Cc1ccc2[nH]cc(C3CNC3)c2c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.41
HTR2C P28335 1/20 0.41
JAK3 P52333 1/20 0.34
OPRD1 P41143 1/20 0.34
OPRK1 P41145 1/20 0.34
HTR1D P28221 2/20 0.33
HTR1B P28222 2/20 0.33
WDR5 P61964 1/20 0.33
MAPK1 P28482 1/20 0.32
CNR1 P21554 1/20 0.32
GABRP O00591 1/20 0.32
GABRD O14764 1/20 0.32
GABRA1 P14867 1/20 0.32
GABRB1 P18505 1/20 0.32
GABRG2 P18507 1/20 0.32
GABRB3 P28472 1/20 0.32
GABRA5 P31644 1/20 0.32
GABRA3 P34903 1/20 0.32
GABRA2 P47869 1/20 0.32
GABRB2 P47870 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7835841 0.81 HTR1A (0.58) HTR1AHTR2COPRK1HTR1DHTR1B
SCHEMBL9545371 0.79 GPR119 (0.40) HTR1AHTR2CJAK3HTR1DHTR1B
SCHEMBL7831800 0.73 HTR1A (0.57) HTR1AHTR2CHTR1DHTR1BCYP2C9
SCHEMBL8784342 0.71 HTR1A (0.53) HTR1AHTR2CHTR1DHTR1BGABRP
SCHEMBL27343955 0.70 HTR1A (0.53) HTR1AHTR2COPRK1HTR1DHTR1B
SCHEMBL21384720 0.65 KDM4E (0.47) HTR1AJAK3OPRK1HTR1DHTR1B
SCHEMBL3713776 0.65 NR1H2 (0.55) NAMPT
SCHEMBL9087213 0.64 HTR1A (0.42) HTR1AHTR2CWDR5FLT3SYK
SCHEMBL9086672 0.64 HTR1A (0.59) HTR1AHTR2CHTR1DHTR1BWDR5
SCHEMBL14211589 0.63 HSD11B1 (0.52) HTR1AHTR1DHTR1BGABRPGABRD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993018029-A1 IMIDAZOLE, TRIAZOLE AND TETRAZOLE DERIVATIVES MERCK SHARP & DOHME LIMITED (GB) 1993-09-16 WO disclosed