SCHEMBL7836166

SCHEMBL7836166

CCOC(=O)CC(CC)NC(=O)CNC(=O)c1cccc(NC(=N)N)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.41
KMT2A Q03164 3/20 0.41
MEN1 O00255 2/20 0.41
GPR139 Q6DWJ6 3/20 0.40
ALDH1A1 P00352 2/20 0.40
F2 P00734 2/20 0.40
F7 P08709 1/20 0.40
PLAU P00749 2/20 0.40
TSHR P16473 2/20 0.40
ITGB3 P05106 1/20 0.39
ITGA2B P08514 1/20 0.39
GAA P10253 1/20 0.39
POLB P06746 1/20 0.39
PKM P14618 1/20 0.39
RAB9A P51151 1/20 0.39
LMNA P02545 2/20 0.38
ALOX15 P16050 1/20 0.38
HTT P42858 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
F10 P00742 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6775429 0.88 ITGB3 (0.44) KMT2AMEN1GPR139ITGB3ITGA2B
SCHEMBL7343613 0.88 KMT2A (0.39) NPSR1KMT2AMEN1GPR139ALDH1A1
SCHEMBL7345100 0.88 NPSR1 (0.43) NPSR1KMT2AMEN1GPR139ALDH1A1
SCHEMBL6779650 0.87 GPR139 (0.43) KMT2AMEN1GPR139ALDH1A1F2
SCHEMBL3839471 0.86 GPR139 (0.47) KMT2AMEN1GPR139F2ITGB3
SCHEMBL7343772 0.86 HTT (0.41) NPSR1KMT2AMEN1GPR139ALDH1A1
SCHEMBL7349391 0.86 ITGB3 (0.56) NPSR1KMT2AMEN1GPR139ALDH1A1
SCHEMBL7349404 0.86 ITGB3 (0.56) NPSR1KMT2AMEN1GPR139ALDH1A1
SCHEMBL7341927 0.86 ITGB3 (0.56) NPSR1KMT2AMEN1GPR139ALDH1A1
SCHEMBL7341726 0.85 GPR139 (0.42) NPSR1KMT2AMEN1GPR139ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0850221-B1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS SEARLE & CO (US) 2001-07-18 EP claimed
CN-1201454-A Meta-guanidino, ureido, thioureido or azacyclic aminobenzoic acid derivatives as integrin antagonists SEARLE & CO (US) 1998-12-09 CN claimed