Phthalylsulfacetamide

Phthalylsulfacetamide

SCHEMBL7836470

CC(=O)NS(=O)(=O)c1ccc(NC(=O)c2ccccc2C(=O)O)cc1.O=C(O)CCC(CCC(=O)O)(C(=O)O)c1ccccc1

nearest known ligand 0.53

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Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.53
MAPT P10636 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.48
HTT P42858 3/20 0.47
PKM P14618 1/20 0.47
CYP3A4 P08684 1/20 0.46
PTGS1 P23219 1/20 0.46
LMNA P02545 1/20 0.46
SCN3A Q9NY46 5/20 0.46
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
HPGD P15428 2/20 0.44
NPC1 O15118 1/20 0.44
TDP1 Q9NUW8 1/20 0.43
HSP90AA1 P07900 1/20 0.43
KDM4E B2RXH2 2/20 0.42
USP2 O75604 1/20 0.42
POLB P06746 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Phthalylsulfacetamide SCHEMBL49529 0.84 ALDH1A1 (0.66) ALDH1A1MAPTL3MBTL1HTTPKM
Phthalylsulfacetamide SCHEMBL3911720 0.83 ALDH1A1 (0.65) ALDH1A1MAPTL3MBTL1HTTPKM
Sulfaloxic Acid SCHEMBL151073 0.71 LMNA (0.56) ALDH1A1MAPTCYP3A4PTGS1LMNA
SCHEMBL27450474 0.71 HSD17B10 (0.71) ALDH1A1MAPTL3MBTL1HTTPKM
SCHEMBL6225889 0.70 ALDH1A1 (0.78) ALDH1A1MAPTL3MBTL1HTTPKM
SCHEMBL18132522 0.69 ALDH1A1 (0.55) ALDH1A1MAPTCYP3A4PTGS1LMNA
SCHEMBL14291632 0.69 ALDH1A1 (0.76) ALDH1A1MAPTL3MBTL1CYP3A4LMNA
SCHEMBL14607436 0.69 ALDH1A1 (0.59) ALDH1A1MAPTL3MBTL1HTTPKM
SCHEMBL11649341 0.69 ALDH1A1 (0.53) ALDH1A1MAPTHTTCYP3A4KDM4E
SCHEMBL18132514 0.68 LMNA (0.72) ALDH1A1MAPTL3MBTL1HTTCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1091958-A1 SALTS OF PAROXETINE SMITHKLINE BEECHAM PLC (GB) 2001-04-18 EP disclosed
WO-2000001692-A1 SALTS OF PAROXETINE SMITHKLINE BEECHAM PLC (GB) 2000-01-13 WO disclosed