SCHEMBL7837858

SCHEMBL7837858

COc1ccccc1Oc1c(Cl)nc(-c2cccs2)nc1NS(=O)(=O)/C=C/c1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.46
HTT P42858 2/20 0.46
EDNRA P25101 6/20 0.41
EDNRB P24530 2/20 0.41
ABCB1 P08183 1/20 0.40
ABCC1 P33527 1/20 0.40
ABCG2 Q9UNQ0 1/20 0.40
DHPS P49366 2/20 0.39
LMNA P02545 3/20 0.39
XPO1 O14980 2/20 0.38
KMT2A Q03164 3/20 0.37
KDM4E B2RXH2 2/20 0.37
MEN1 O00255 2/20 0.37
MAPT P10636 2/20 0.37
MAPK1 P28482 2/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
NFE2L2 Q16236 2/20 0.37
PKM P14618 1/20 0.36
HPGD P15428 1/20 0.36
GBA1 P04062 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7837861 1.00 ALDH1A1 (0.46) ALDH1A1HTTEDNRAEDNRBABCB1
SCHEMBL7837700 0.90 ALDH1A1 (0.47) ALDH1A1HTTEDNRAEDNRBABCB1
SCHEMBL7837698 0.90 ALDH1A1 (0.47) ALDH1A1HTTEDNRAEDNRBABCB1
SCHEMBL7844686 0.87 DHPS (0.54) ALDH1A1HTTEDNRAEDNRBDHPS
SCHEMBL7844683 0.87 DHPS (0.54) ALDH1A1HTTEDNRAEDNRBDHPS
SCHEMBL7839633 0.85 EDNRA (0.50) ALDH1A1HTTEDNRAEDNRBDHPS
SCHEMBL7839629 0.85 EDNRA (0.50) ALDH1A1HTTEDNRAEDNRBDHPS
SCHEMBL5271698 0.85 EDNRA (0.52) ALDH1A1HTTEDNRAEDNRB
SCHEMBL5271700 0.85 EDNRA (0.52) ALDH1A1HTTEDNRAEDNRB
SCHEMBL7840781 0.85 ALDH1A1 (0.45) ALDH1A1HTTEDNRAEDNRBDHPS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0882719-B1 ARYLETHENESULFONAMIDE DERIVATIVES AND DRUG COMPOSITION CONTAINING THE SAME YAMANOUCHI PHARMA CO LTD (JP) 2001-05-16 EP disclosed
US-6083955-A HAVING A HIGH AFFINITY FOR DRUGS, ESPECIALLY ENDOSERINE RECEPTORS YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 2000-07-04 US disclosed
EP-0882719-A1 ARYLETHENESULFONAMIDE DERIVATIVES AND DRUG COMPOSITION CONTAINING THE SAME YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1998-12-09 EP disclosed