SCHEMBL7838129

SCHEMBL7838129

O=C1Cc2ccccc2CCc2ccccc21

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 2/20 0.60
CYP2A6 P11509 2/20 0.59
MAOA P21397 2/20 0.59
MAOB P27338 2/20 0.59
BCHE P06276 1/20 0.56
ALDH1A1 P00352 4/20 0.52
KDM4E B2RXH2 3/20 0.52
HPGD P15428 2/20 0.52
CYP1A2 P05177 1/20 0.48
PDPK1 O15530 1/20 0.45
PARP1 P09874 1/20 0.45
PARP10 Q53GL7 1/20 0.45
PARP11 Q9NR21 1/20 0.45
TDP1 Q9NUW8 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
CYP3A4 P08684 1/20 0.43
MAPT P10636 1/20 0.43
PABPC1 P11940 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31392106 0.86 CES1 (0.67) CES1CYP2A6MAOAMAOBBCHE
SCHEMBL3638469 0.86 CES1 (0.67) CES1CYP2A6MAOAMAOBBCHE
SCHEMBL31070117 0.85
SCHEMBL569873 0.85
SCHEMBL8035811 0.85 CES1 (0.73) CES1CYP2A6MAOAMAOBBCHE
SCHEMBL29353311 0.83 MAOA (0.74) CES1CYP2A6MAOAMAOBBCHE
SCHEMBL1268680 0.83 MAOA (0.74) CES1CYP2A6MAOAMAOBBCHE
SCHEMBL24746 0.83 MAOA (0.74) CES1CYP2A6MAOAMAOBBCHE
SCHEMBL31454252 0.81 MAOA (0.71) CES1CYP2A6MAOAMAOBBCHE
Bromide SCHEMBL28903594 0.81 MAOA (0.71) CES1CYP2A6MAOAMAOBBCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170320815-A1 ALKYNES AND METHODS OF REACTING ALKYNES WITH 1,3-DIPOLE-FUNCTIONAL COMPOUNDS UNIVERSITY OF GEORGIA RESEARCH FOUNDATION, INC. 2017-11-09 US disclosed
US-7582667-B2 Dihydrospiro[dibenzo[a,d][7]annulene-5,4′-imidazol] compounds for the inhibition of beta-secretase WYETH (US) 2009-09-01 US disclosed
US-20070203116-A1 Dihydrospiro[dibenzo[a,d][7]annulene-5,4'-imidazol] compounds for the inhibition of beta-secretase WYETH (US) 2007-08-30 US disclosed
EP-0820450-B1 N-substituted azaheterocyclic carboxylic acids and alkylesters thereof NOVO NORDISK AS (DK) 2001-09-12 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170320815-A1 ALKYNES AND METHODS OF REACTING ALKYNES WITH 1,3-DIPOLE-FUNCTIONAL COMPOUNDS ALG1, ST3GAL3, B3GNT2 CES1 2397/4885CYP2A6 2372/4885MAOA 270/4885
US-20070203116-A1 Dihydrospiro[dibenzo[a,d][7]annulene-5,4'-imidazol] compounds for the inhibition of beta-secretase BACE1, BACE2, APP CES1 880/4885CYP2A6 4102/4885MAOA 658/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.