SCHEMBL7840653

SCHEMBL7840653

c1ccc(CN2CCC(Nc3ccccc3-c3ccccc3)CC2)cc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.68
KDM4E B2RXH2 1/20 0.68
MAPK1 P28482 2/20 0.61
ACHE P22303 6/20 0.57
BCHE P06276 4/20 0.56
MALT1 Q9UDY8 1/20 0.56
BACE1 P56817 3/20 0.56
ROCK2 O75116 2/20 0.56
ROCK1 Q13464 1/20 0.56
MAPT P10636 3/20 0.55
KMT2A Q03164 3/20 0.55
NPSR1 Q6W5P4 2/20 0.55
MEN1 O00255 2/20 0.55
ALDH1A1 P00352 2/20 0.55
LMNA P02545 1/20 0.54
NTSR1 P30989 1/20 0.54
HTT P42858 1/20 0.54
PKM P14618 1/20 0.52
RAB9A P51151 1/20 0.52
SIGMAR1 Q99720 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7007839 0.85 KDM4E (0.64) GAAKDM4EMAPK1ACHEBCHE
SCHEMBL7286176 0.82 KDM4E (0.67) GAAKDM4EMAPK1ACHEBCHE
SCHEMBL7289451 0.81 KDM4E (0.70) GAAKDM4EMAPK1ACHEBCHE
SCHEMBL28332709 0.81 KDM4E (0.70) GAAKDM4EMAPK1ACHEBCHE
SCHEMBL5671677 0.81 KDM4E (0.70) GAAKDM4EMAPK1ACHEBCHE
SCHEMBL13717362 0.81 SIGMAR1 (0.70) GAAKDM4EMAPK1MAPTKMT2A
SCHEMBL13718274 0.81 ALDH1A1 (0.57) GAAKDM4EMAPK1MAPTKMT2A
Hydrochloric Acid SCHEMBL11102409 0.80 KDM4E (0.68) GAAKDM4EMAPK1ACHEBCHE
SCHEMBL7014000 0.80 MAPK1 (0.82) GAAKDM4EMAPK1ACHEBCHE
SCHEMBL29127243 0.79 ALDH1A1 (0.49) GAAKDM4EMAPTKMT2ANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1163239-A1 MODIFIED AMINO-ACID AMIDES AS CGRP ANTAGONISTS Boehringer Ingelheim Pharma KG (DE) 2001-12-19 EP disclosed
WO-2000055154-A1 MODIFIED AMINO-ACID AMIDES AS CGRP ANTAGONISTS BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-09-21 WO disclosed