SCHEMBL7840693

SCHEMBL7840693

O=[N+]([O-])c1cc(CCNCc2ccccc2)ccc1OCc1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.57
SLC2A1 P11166 1/20 0.56
BCHE P06276 5/20 0.54
PDCD1 Q15116 4/20 0.54
CD274 Q9NZQ7 4/20 0.54
POLB P06746 2/20 0.54
KCNH2 Q12809 1/20 0.54
MEN1 O00255 3/20 0.53
KMT2A Q03164 3/20 0.53
ALDH1A1 P00352 3/20 0.53
CTSV O60911 1/20 0.52
CTSL P07711 1/20 0.52
SMN1; SMN2 Q16637 2/20 0.51
LMNA P02545 1/20 0.51
HTT P42858 1/20 0.51
GAA P10253 1/20 0.50
CA12 O43570 1/20 0.50
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
CA9 Q16790 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11669913 0.99 KDM4E (0.56) KDM4ESLC2A1BCHEPDCD1CD274
Bromide SCHEMBL11670771 0.99 KDM4E (0.56) KDM4ESLC2A1BCHEPDCD1CD274
SCHEMBL4643754 0.90 CTSV (0.56) KDM4EBCHEPDCD1CD274POLB
SCHEMBL10646744 0.84 ALDH1A1 (0.51) KDM4EPDCD1CD274POLBMEN1
SCHEMBL3599069 0.82 POLB (0.54) POLBMEN1KMT2AALDH1A1CTSV
SCHEMBL5642071 0.82 CTSV (0.56) PDCD1CD274POLBMEN1KMT2A
SCHEMBL6814063 0.82 POLB (0.54) PDCD1CD274POLBMEN1KMT2A
SCHEMBL7279743 0.82 SLC2A1 (0.80) KDM4ESLC2A1BCHEMEN1KMT2A
SCHEMBL6235952 0.81 PDCD1 (0.51) KDM4ESLC2A1BCHEPDCD1CD274
Hydrochloric Acid SCHEMBL7839532 0.81 POLB (0.53) POLBMEN1KMT2AALDH1A1CTSV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0558677-B1 BIOLOGICALLY ACTIVE AMINES ASTRAZENECA AB (SE) 2001-08-16 EP disclosed
US-5763465-A 7-(2-aminoethyl) benzothiazolones ASTRA PHARMACEUTICALS LIMITED (GB) 1998-06-09 US disclosed
US-5648370-A 7-(2-aminoethyl) benzothiazolones ASTRA PHARMACEUTICALS LIMITED (GB) 1997-07-15 US disclosed
WO-1992008708-A1 BIOLOGICALLY ACTIVE AMINES FISONS PLC (GB) 1992-05-29 WO disclosed
US-4024281-A N,N-bis[2-(3-substituted-4-hydroxyphenyl)-ethyl or -2-hydroxyethyl]-polymethylenediamines SMITHKLINE CORPORATION (US) 1977-05-17 US disclosed
US-3933913-A N,N'-bis[3-substituted-4-hydroxypheyl)-2-hydroxyethyl)]-polymethylenediamines SMITHKLINE CORPORATION (US) 1976-01-20 US disclosed