SCHEMBL7841369

SCHEMBL7841369

COC(=O)c1ncc(C)c(C)c1N

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.42
TSHR P16473 1/20 0.39
KDM4E B2RXH2 7/20 0.38
ALDH1A1 P00352 6/20 0.38
GAA P10253 3/20 0.38
MAPK1 P28482 2/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
GLA P06280 2/20 0.38
HSD17B10 Q99714 4/20 0.37
HPGD P15428 3/20 0.37
CYP3A4 P08684 1/20 0.36
ACHE P22303 1/20 0.36
ATM Q13315 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
TP53 P04637 1/20 0.36
CASP1 P29466 1/20 0.35
HTT P42858 1/20 0.35
CASP7 P55210 1/20 0.35
NCOA1 Q15788 1/20 0.35
RCE1 Q9Y256 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21072556 0.75 NOS3 (0.47) NPSR1KDM4EALDH1A1GAAMAPK1
SCHEMBL5820179 0.75 NPSR1 (0.42) NPSR1TSHRKDM4EALDH1A1GAA
SCHEMBL22439846 0.75 NPSR1 (0.47) NPSR1TSHRKDM4EALDH1A1GAA
SCHEMBL7665937 0.75 AGXT (0.44) NPSR1TSHRKDM4EALDH1A1MAPK1
SCHEMBL1840938 0.73 NPSR1 (0.43) NPSR1TSHRKDM4EALDH1A1GAA
SCHEMBL289542 0.71 OPRK1 (0.44) NPSR1ATM
SCHEMBL18124754 0.71 ATM (0.47) NPSR1TSHRKDM4EALDH1A1GAA
SCHEMBL12248189 0.71 NPSR1 (0.47) NPSR1TSHRKDM4EALDH1A1GAA
SCHEMBL26684922 0.71 NPSR1 (0.38) NPSR1TSHRKDM4EALDH1A1GAA
SCHEMBL25581894 0.70 NPSR1 (0.50) NPSR1KDM4EALDH1A1GAAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0805812-B1 BICYCLIC SUBSTITUTED HEXAHYDROBENZ(E)ISOINDOLE ALPHA-1- ADRENERGIC ANTAGONISTS ABBOTT LAB (US) 2001-06-13 EP disclosed
US-5792767-A TREATMENT OF BENIGN PROSTATIC HYPERTROPY ABBOTT LABORATORIES (US) 1998-08-11 US disclosed