SCHEMBL7841948

SCHEMBL7841948

CC(=O)C(=C(C(=O)O)c1ccc(Cl)cc1)c1ccccc1S(C)(=O)=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCAT2 O15382 1/20 0.44
NR4A1 P22736 1/20 0.42
AKR1C3 P42330 2/20 0.40
CES2 O00748 1/20 0.40
CES1 P23141 1/20 0.40
AKR1C2 P52895 1/20 0.40
AKR1C1 Q04828 1/20 0.40
PTGS2 P35354 1/20 0.40
LMNA P02545 2/20 0.40
MEN1 O00255 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C19 P33261 1/20 0.39
KMT2A Q03164 1/20 0.39
HSD11B1 P28845 2/20 0.38
CYP19A1 P11511 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
RAB9A P51151 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7840110 0.86 BCAT2 (0.40) BCAT2NR4A1AKR1C3AKR1C2AKR1C1
SCHEMBL7844137 0.86 BCAT2 (0.44) BCAT2AKR1C3AKR1C2AKR1C1PTGS2
SCHEMBL7641541 0.80 AKR1C3 (0.57) AKR1C3AKR1C2AKR1C1PTGS2
SCHEMBL7641537 0.80 AKR1C3 (0.57) AKR1C3AKR1C2AKR1C1PTGS2
SCHEMBL13776409 0.80 AKR1C3 (0.57) AKR1C3AKR1C2AKR1C1PTGS2
SCHEMBL8002389 0.78 BCAT2 (0.50) BCAT2CES2CES1AKR1C2AKR1C1
SCHEMBL6250243 0.78 BCAT2 (0.50) BCAT2CES2CES1AKR1C2AKR1C1
SCHEMBL7829901 0.73 BCAT2 (0.40) BCAT2AKR1C3AKR1C2AKR1C1PTGS2
SCHEMBL34748 0.69 BCAT2 (0.62) BCAT2LMNAKDM4EALDH1A1
SCHEMBL30455577 0.69 BCAT2 (0.62) BCAT2LMNAMEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0828724-B1 DIARYL-5-OXYGENATED-2-(5H)-FURANONES AS COX-2 INHIBITORS MERCK FROSST CANADA INC (CA) 2001-12-05 EP claimed