SCHEMBL7999933

SCHEMBL7999933

N#Cc1c(Nc2ccccc2)nc2ccccc2c1CCc1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.51
KMT2A Q03164 5/20 0.51
NPSR1 Q6W5P4 1/20 0.51
RXFP1 Q9HBX9 1/20 0.51
ALDH1A1 P00352 4/20 0.46
KDM4E B2RXH2 3/20 0.44
MAPT P10636 2/20 0.43
LMNA P02545 2/20 0.43
TP53 P04637 1/20 0.43
CYP1A2 P05177 1/20 0.43
TSHR P16473 1/20 0.43
HSD17B10 Q99714 1/20 0.43
ABCG2 Q9UNQ0 5/20 0.42
NPY5R Q15761 1/20 0.42
PDE5A O76074 2/20 0.41
ADORA2A P29274 1/20 0.40
ADORA1 P30542 1/20 0.40
KDM1A O60341 1/20 0.40
DAPK3 O43293 1/20 0.39
MAP4K4 O95819 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7845574 0.79 MEN1 (0.48) MEN1KMT2ANPSR1RXFP1ALDH1A1
SCHEMBL6071945 0.78 ALDH1A1 (0.49) MEN1KMT2ANPSR1RXFP1ALDH1A1
SCHEMBL7826836 0.77 MEN1 (0.45) MEN1KMT2ANPSR1RXFP1ALDH1A1
SCHEMBL20259096 0.76 ALDH1A1 (0.58) MEN1KMT2ANPSR1RXFP1ALDH1A1
SCHEMBL7689600 0.76 ALDH1A1 (0.51) MEN1KMT2ANPSR1RXFP1ALDH1A1
SCHEMBL7836872 0.75 MEN1 (0.45) MEN1KMT2ANPSR1RXFP1ALDH1A1
SCHEMBL7842318 0.75 MEN1 (0.47) MEN1KMT2ANPSR1RXFP1ALDH1A1
SCHEMBL7999981 0.75 MEN1 (0.45) MEN1KMT2ANPSR1RXFP1ALDH1A1
SCHEMBL7999931 0.70 ALDH1A1 (0.48) MEN1KMT2ANPSR1RXFP1ALDH1A1
SCHEMBL7999926 0.70 MEN1 (0.50) MEN1KMT2ANPSR1RXFP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6288082-B1 COMPOUNDS SUCH AS 6,7-DIETHOXY-4-(INDAN-5-YLAMINO) -QUINOLINE-3-CARBONITRILE USED AS ANTINEOPLASTIC AGENTS AND IN THE TREATMENT OF POLYCYCSTIC KIDNEY DISEASE AMERICAN CYANAMID COMPANY 2001-09-11 US disclosed