SCHEMBL7851328

SCHEMBL7851328

Cc1nc2[nH]cc(C#Cc3ccc(C(=O)O)s3)c2c(=O)[nH]1

nearest known ligand 0.33

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DAO P14920 1/20 0.33
LMNA P02545 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
TYMS P04818 2/20 0.32
ALDH1A1 P00352 1/20 0.32
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32
KDM4C Q9H3R0 1/20 0.32
MAPK1 P28482 1/20 0.32
PARP1 P09874 1/20 0.31
FOLR1 P15328 4/20 0.31
SLC19A1 P41440 3/20 0.31
SLC46A1 Q96NT5 3/20 0.31
ADORA3 P0DMS8 1/20 0.30
ADORA2A P29274 1/20 0.30
GART P22102 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7854494 0.78 TYMS (0.43) TYMSGAA
SCHEMBL7841320 0.73 DAO (0.36) DAOLMNAL3MBTL1TYMSALDH1A1
SCHEMBL7842455 0.72 PARP1 (0.36) L3MBTL1TYMSALDH1A1MAPK1PARP1
SCHEMBL26232174 0.70 CHUK (0.49) GAA
SCHEMBL22071237 0.68 DAO (0.52) DAOL3MBTL1ALDH1A1GAA
SCHEMBL17057395 0.65 DAO (0.43) DAOL3MBTL1ALDH1A1GAAMAPT
SCHEMBL26232177 0.64 TYMS (0.41) L3MBTL1TYMSALDH1A1MAPK1PARP1
SCHEMBL7851196 0.62 TYMS (0.48) L3MBTL1TYMSALDH1A1MAPK1PARP1
SCHEMBL4407685 0.60 RAB9A (0.44) DAOL3MBTL1ALDH1A1
SCHEMBL17053135 0.60 FFAR1 (0.50) DAOL3MBTL1ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0923287-A4 NONCLASSICAL PYRROLO 2,3-D]PYRIMIDINE ANTIFOLATES LILLY CO ELI (US) 2001-08-01 EP disclosed
EP-0923287-A1 NONCLASSICAL PYRROLO 2,3-D]PYRIMIDINE ANTIFOLATES ELI LILLY AND COMPANY (US) 1999-06-23 EP disclosed
WO-1998008382-A1 NONCLASSICAL PYRROLO[2,3-D]PYRIMIDINE ANTIFOLATES ELI LILLY AND COMPANY (US) 1998-03-05 WO disclosed