SCHEMBL7842482

SCHEMBL7842482

CS(=O)(=O)c1ccc(-c2sc(C(=O)NCc3cccc(F)c3)nc2-c2ccc(F)cc2)cc1

nearest known ligand 0.59

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 18/20 0.59
PTGS1 P23219 2/20 0.55
MAOB P27338 1/20 0.52
ROCK2 O75116 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7843450 1.00 PTGS2 (0.59) PTGS2PTGS1MAOBROCK2
SCHEMBL7844757 0.92 PTGS2 (0.56) PTGS2PTGS1
SCHEMBL7844442 0.92 PTGS2 (0.56) PTGS2PTGS1
SCHEMBL7844808 0.92 PTGS2 (0.56) PTGS2PTGS1MAOB
SCHEMBL7843264 0.92 PTGS2 (0.56) PTGS2PTGS1MAOB
SCHEMBL7844196 0.91 PTGS2 (0.62) PTGS2PTGS1
SCHEMBL7832863 0.91 PTGS2 (0.62) PTGS2PTGS1
SCHEMBL7841076 0.91 PTGS2 (0.66) PTGS2PTGS1
SCHEMBL7846333 0.91 PTGS2 (0.66) PTGS2PTGS1
SCHEMBL7841669 0.90 MAOB (0.52) PTGS2PTGS1MAOBROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1125932-A2 Substituted thiazoles for the treatment of inflammation G.D. SEARLE & CO. (US) 2001-08-22 EP disclosed
US-5668161-A Substituted thiazoles for the treatment of inflammation G.D. SEARLE & CO. (US) 1997-09-16 US disclosed
EP-0772606-A1 SUBSTITUTED THIAZOLES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1997-05-14 EP disclosed
WO-1996003392-A1 SUBSTITUTED THIAZOLES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-02-08 WO disclosed