SCHEMBL7842583

SCHEMBL7842583

[NH]C(=O)C(CCN)N1CCNCC1

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.38
OPRD1 P41143 2/20 0.32
CHRM5 P08912 1/20 0.31
CHRM3 P20309 1/20 0.31
CA12 O43570 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
CA9 Q16790 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1401532 0.84 SIGMAR1 (0.38) SIGMAR1OPRD1
SCHEMBL2764645 0.84 SIGMAR1 (0.38) SIGMAR1OPRD1CHRM5CHRM3CA12
SCHEMBL8387444 0.71 GSR (0.42) SIGMAR1
SCHEMBL28958643 0.70 OPRD1 (0.40) SIGMAR1OPRD1CHRM5CHRM3CA12
SCHEMBL30903250 0.70 SLC6A4 (0.41)
SCHEMBL8310688 0.69 SIGMAR1 (0.41) SIGMAR1OPRD1CHRM5CHRM3CA12
SCHEMBL1077282 0.69 SIGMAR1 (0.38) SIGMAR1OPRD1CHRM5CHRM3CA12
SCHEMBL28252629 0.68 SLC6A4 (0.37)
SCHEMBL1905214 0.68 SIGMAR1 (0.47) SIGMAR1CA12CA1CA2CA9
SCHEMBL9801277 0.67 SLC6A4 (0.32) SIGMAR1CHRM5CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1071668-A1 5-AMINOINDENO(1,2-C)PYRAZOL-4-ONES AS ANTI-CANCER AND ANTI-PROLIFERATIVE AGENTS Du Pont Pharmaceuticals Company (US) 2001-01-31 EP disclosed
WO-1999054308-A1 5-AMINOINDENO(1,2-C)PYRAZOL-4-ONES AS ANTI-CANCER AND ANTI-PROLIFERATIVE AGENTS DU PONT PHARMACEUTICALS COMPANY (US) 1999-10-28 WO disclosed