SCHEMBL7842750

SCHEMBL7842750

COc1ccccc1Oc1c(Cl)nc(-c2ccc(C(F)(F)F)nc2)nc1NS(=O)(=O)/C=C/c1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DHPS P49366 8/20 0.42
ALDH1A1 P00352 1/20 0.42
HTT P42858 1/20 0.42
EDNRA P25101 10/20 0.41
EDNRB P24530 5/20 0.40
SCN9A Q15858 1/20 0.39
ABCC3 O15438 1/20 0.38
ABCC4 O15439 1/20 0.38
NR1I2 O75469 1/20 0.38
ABCB11 O95342 1/20 0.38
NR1H3 Q13133 1/20 0.38
NR1I3 Q14994 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7842752 1.00 DHPS (0.42) DHPSALDH1A1HTTEDNRAEDNRB
SCHEMBL7840308 0.91 EDNRA (0.47) DHPSALDH1A1HTTEDNRAEDNRB
SCHEMBL7840305 0.91 EDNRA (0.47) DHPSALDH1A1HTTEDNRAEDNRB
SCHEMBL7840415 0.89 ALDH1A1 (0.45) DHPSALDH1A1HTTEDNRAEDNRB
SCHEMBL7840413 0.89 ALDH1A1 (0.45) DHPSALDH1A1HTTEDNRAEDNRB
SCHEMBL7842387 0.88 DHPS (0.47) DHPSALDH1A1HTTEDNRAEDNRB
SCHEMBL7842383 0.88 DHPS (0.47) DHPSALDH1A1HTTEDNRAEDNRB
SCHEMBL7844463 0.87 EDNRA (0.58) DHPSEDNRAEDNRBABCC3ABCC4
SCHEMBL7844466 0.87 EDNRA (0.58) DHPSEDNRAEDNRBABCC3ABCC4
SCHEMBL7844686 0.86 DHPS (0.54) DHPSALDH1A1HTTEDNRAEDNRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0882719-B1 ARYLETHENESULFONAMIDE DERIVATIVES AND DRUG COMPOSITION CONTAINING THE SAME YAMANOUCHI PHARMA CO LTD (JP) 2001-05-16 EP disclosed
US-6083955-A HAVING A HIGH AFFINITY FOR DRUGS, ESPECIALLY ENDOSERINE RECEPTORS YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 2000-07-04 US disclosed
EP-0882719-A1 ARYLETHENESULFONAMIDE DERIVATIVES AND DRUG COMPOSITION CONTAINING THE SAME YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1998-12-09 EP disclosed