SCHEMBL78430

SCHEMBL78430

COCCCn1ncc2ccc(C(C)C)cc21

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
REN P00797 2/20 0.50
MAPK1 P28482 2/20 0.47
HTR2A P28223 5/20 0.44
HTR2C P28335 5/20 0.44
HTR2B P41595 4/20 0.44
KMO O15229 5/20 0.40
HTR1A P08908 2/20 0.40
ADRA2A P08913 2/20 0.40
ADRA2B P18089 2/20 0.40
ADRA2C P18825 2/20 0.40
HTR1D P28221 1/20 0.40
HTR7 P34969 1/20 0.40
HTR4 Q13639 1/20 0.40
CHRM2 P08172 3/20 0.40
CHRM1 P11229 3/20 0.40
CHRM3 P20309 2/20 0.40
CASR P41180 1/20 0.38
MEN1 O00255 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16471691 0.82 REN (0.50) RENMAPK1HTR2AHTR2CHTR2B
SCHEMBL15417971 0.82 MAPK1 (0.59) RENMAPK1HTR2AHTR2CHTR2B
SCHEMBL91363 0.82 KMO (0.58) RENMAPK1HTR2AHTR2CHTR2B
SCHEMBL19697957 0.81 HTR2A (0.44) MAPK1HTR2AHTR2CHTR2BKMO
SCHEMBL29305629 0.81 MAOB (0.49) MAPK1HTR2AHTR2CHTR2BKMO
SCHEMBL3779615 0.81 KMO (0.42) RENMAPK1HTR2AHTR2CHTR2B
SCHEMBL3777719 0.81 HTR2A (0.44) RENMAPK1HTR2AHTR2CHTR2B
SCHEMBL3086407 0.80 KMO (0.44) RENMAPK1HTR2AHTR2CHTR2B
SCHEMBL3074398 0.78 KMO (0.43) RENMAPK1HTR2AHTR2CHTR2B
SCHEMBL3780833 0.78 KMO (0.40) RENMAPK1HTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed