SCHEMBL7843059

SCHEMBL7843059

CC(C)(C)OC(=O)Nc1nc(CC(=O)Nc2nc(CC(=O)O)cs2)cs1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.53
SMN1; SMN2 Q16637 3/20 0.53
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53
HPGD P15428 1/20 0.53
POLB P06746 2/20 0.49
GAA P10253 2/20 0.48
ITGB1 P05556 1/20 0.47
ITGA4 P13612 1/20 0.47
PDE5A O76074 3/20 0.47
SLC12A2 P55011 1/20 0.47
SLC12A5 Q9H2X9 1/20 0.47
KDM4E B2RXH2 2/20 0.47
SIRT1 Q96EB6 1/20 0.46
ESR2 Q92731 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL299175 0.95 SMN1; SMN2 (0.51) ALDH1A1SMN1; SMN2MEN1KMT2AHPGD
Trifluoromethanesulfonic Acid SCHEMBL29356486 0.86 ALDH1A1 (0.44) ALDH1A1SMN1; SMN2POLBGAASIRT1
SCHEMBL8177534 0.84 ALDH1A1 (0.45) ALDH1A1SMN1; SMN2MEN1KMT2AHPGD
SCHEMBL9727370 0.84 SMN1; SMN2 (0.51) ALDH1A1SMN1; SMN2MEN1KMT2AHPGD
SCHEMBL7419507 0.83 SMN1; SMN2 (0.56) ALDH1A1SMN1; SMN2MEN1KMT2AHPGD
SCHEMBL29557286 0.83 SIRT1 (0.53) ALDH1A1SMN1; SMN2MEN1KMT2AHPGD
SCHEMBL774746 0.82 LCK (0.55) ALDH1A1SMN1; SMN2HPGDGAAPDE5A
SCHEMBL1030124 0.81 PI4KB (0.50) ALDH1A1SMN1; SMN2KMT2AHPGDGAA
SCHEMBL2175797 0.81 SMN1; SMN2 (0.50) ALDH1A1SMN1; SMN2KMT2AHPGDGAA
SCHEMBL5481490 0.81 CCNE1 (0.51) ALDH1A1SMN1; SMN2MEN1KMT2AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0984963-B1 NOVEL COMPOUNDS ASTRAZENECA AB (SE) 2001-04-11 EP disclosed
US-6162808-A Compounds ASTRAZENECA U.K. LIMITED (GB) 2000-12-19 US disclosed