SCHEMBL7843213

SCHEMBL7843213

CCOC(=O)CN(C)C(=O)c1ccc(C(=O)c2cccnc2C(=O)N(C)CC(=O)OCC)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.39
MAPT P10636 2/20 0.39
BRD4 O60885 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
HTT P42858 1/20 0.38
MAPK1 P28482 1/20 0.38
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38
NPC1 O15118 3/20 0.37
RAB9A P51151 3/20 0.37
HPGD P15428 1/20 0.37
KDM4E B2RXH2 1/20 0.37
GAA P10253 1/20 0.37
ALOX15 P16050 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
LMNA P02545 1/20 0.37
PDK1 Q15118 1/20 0.37
PDK2 Q15119 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7850370 0.83 L3MBTL1 (0.47) ALDH1A1MAPTTDP1HTTMAPK1
SCHEMBL1921859 0.81 BRD4 (0.42) ALDH1A1MAPTBRD4HTTCA12
SCHEMBL7853990 0.79 L3MBTL1 (0.44) ALDH1A1MAPTNPC1RAB9AHPGD
SCHEMBL19017656 0.78 CYP2C19 (0.47) ALDH1A1MAPTTDP1SMN1; SMN2LMNA
SCHEMBL7851483 0.77 MAPT (0.40) ALDH1A1MAPTCA12CA1CA2
SCHEMBL7851482 0.75 COMT (0.43) ALDH1A1MAPTTDP1NPC1RAB9A
SCHEMBL30038114 0.75 HTT (0.50) ALDH1A1MAPTHTTMAPK1KDM4E
SCHEMBL14679109 0.74 CA12 (0.51) ALDH1A1MAPTTDP1CA12CA1
SCHEMBL7852266 0.74 COMT (0.41) ALDH1A1TDP1NPC1RAB9AHPGD
SCHEMBL8785261 0.74 LMNA (0.46) MAPTCA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0652218-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2001-07-11 EP disclosed
US-5585385-A USEFUL IN TREATING DISORDERS OF MICTURITION; ADMINISTERING TO INHIBIT PLASMA EXTRAVASATION TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-12-17 US disclosed