SCHEMBL7843260

SCHEMBL7843260

CCOC(=O)c1c(-c2ccc(F)cc2)c2ccn(C)c2c(=O)n1C

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GABRA2 P47869 1/20 0.41
GABRB2 P47870 1/20 0.41
MAPT P10636 5/20 0.41
MEN1 O00255 4/20 0.41
KMT2A Q03164 4/20 0.41
CASP3 P42574 1/20 0.41
TRPV1 Q8NER1 1/20 0.41
SENP7 Q9BQF6 1/20 0.41
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
GAA P10253 1/20 0.39
HPGD P15428 1/20 0.39
CENPE Q02224 2/20 0.39
CHRNA7 P36544 1/20 0.39
TSHR P16473 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
GPR55 Q9Y2T6 1/20 0.38
TACR1 P25103 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8989478 0.84 CENPE (0.53) GABRA2GABRB2MAPTMEN1KMT2A
SCHEMBL7851323 0.83 GRIA4 (0.44) CENPETACR1
SCHEMBL7852329 0.79 TP53 (0.41) GABRA2GABRB2MAPTMEN1KMT2A
SCHEMBL5233063 0.78 TACR1 (0.46) KDM4EALDH1A1HPGDCENPETSHR
SCHEMBL7853648 0.78 MAPK14 (0.44) GABRA2GABRB2MAPTMEN1KMT2A
SCHEMBL7850580 0.78 MAPK14 (0.44) GABRA2GABRB2MAPTMEN1KMT2A
SCHEMBL27364098 0.77 TP53 (0.35) MAPTMEN1KMT2AALDH1A1CENPE
SCHEMBL9301200 0.76 ELANE (0.53) GABRA2GABRB2MAPTMEN1KMT2A
SCHEMBL7851659 0.76 TACR1 (0.46) GABRA2GABRB2MAPTKDM4EALDH1A1
SCHEMBL14809648 0.75 MEN1 (0.42) MAPTMEN1KMT2AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0652218-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2001-07-11 EP disclosed
CN-1052004-C Heterocyclic compounds, their production and use TALCEDA CHEMICAL IND LTD (JP) 2000-05-03 CN disclosed
US-5585385-A USEFUL IN TREATING DISORDERS OF MICTURITION; ADMINISTERING TO INHIBIT PLASMA EXTRAVASATION TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-12-17 US disclosed
CN-1107476-A Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1995-08-30 CN disclosed
EP-0652218-A1 Heterocyclic compounds, their production and use Takeda Chemical Industries, Ltd. (JP) 1995-05-10 EP disclosed