SCHEMBL7843354

SCHEMBL7843354

CC(C)=CCc1cc(C#N)ccc1Br

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARG P37231 1/20 0.38
PPARA Q07869 1/20 0.38
HTT P42858 3/20 0.36
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
TTR P02766 1/20 0.35
ALB P02768 1/20 0.35
HPGD P15428 2/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
PTGS1 P23219 1/20 0.34
PTGS2 P35354 1/20 0.34
ALDH1A1 P00352 1/20 0.34
SETDB1 Q15047 1/20 0.34
AKR1B10 O60218 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7505085 0.79 CYP2A6 (0.32) HTTMEN1KMT2ATTRALB
SCHEMBL2934457 0.75 CYP2A6 (0.47) MEN1KMT2ATTRALBALDH1A1
SCHEMBL500133 0.75 MEN1 (0.42) MEN1KMT2ATTRALBPTPN1
SCHEMBL1232330 0.73 MEN1 (0.39) HTTMEN1KMT2ATTRALB
SCHEMBL20482939 0.73 MEN1 (0.39) MEN1KMT2ATTRALBPTPN1
SCHEMBL4773225 0.73 MEN1 (0.43) MEN1KMT2ATTRALBALDH1A1
SCHEMBL1232549 0.72 ALDH1A1 (0.38) KMT2ACYP3A4ALDH1A1SETDB1CXCR1
SCHEMBL27528549 0.72 LOXL2 (0.47) HTTMEN1KMT2ATTRALB
SCHEMBL4774237 0.71 ALDH1A1 (0.37) MEN1KMT2ATTRALBHPGD
SCHEMBL8536839 0.71 MAOB (0.37) MEN1KMT2ATTRALBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1094816-A4 BIPHENYL SULFONAMIDES AS DUAL ANGIOTENSIN ENDOTHELIN RECEPTOR ANTAGONISTS BRISTOL MYERS SQUIBB CO (US) 2001-12-19 EP disclosed
EP-1094816-A1 BIPHENYL SULFONAMIDES AS DUAL ANGIOTENSIN ENDOTHELIN RECEPTOR ANTAGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2001-05-02 EP disclosed
WO-2000001389-A1 BIPHENYL SULFONAMIDES AS DUAL ANGIOTENSIN ENDOTHELIN RECEPTOR ANTAGONISTS BRISTOL-MYERS SQUIBB CO. (US) 2000-01-13 WO disclosed