SCHEMBL7843519

SCHEMBL7843519

COc1ccccc1Oc1c(Cl)nc(-c2cccnc2)nc1NS(=O)(=O)/C=C/c1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.46
KMT2A Q03164 4/20 0.46
MAPT P10636 3/20 0.46
GAA P10253 2/20 0.46
MEN1 O00255 2/20 0.46
NPSR1 Q6W5P4 1/20 0.46
DHPS P49366 5/20 0.45
HTT P42858 1/20 0.45
EDNRA P25101 5/20 0.44
EDNRB P24530 4/20 0.44
MAPK1 P28482 2/20 0.42
KDM4E B2RXH2 2/20 0.42
POLB P06746 1/20 0.42
RECQL P46063 1/20 0.42
LMNA P02545 2/20 0.41
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 2/20 0.41
GMNN O75496 1/20 0.41
ADORA3 P0DMS8 1/20 0.41
ADORA2B P29275 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7843522 1.00 ALDH1A1 (0.46) ALDH1A1KMT2AMAPTGAAMEN1
SCHEMBL7844686 0.92 DHPS (0.54) ALDH1A1DHPSHTTEDNRAEDNRB
SCHEMBL7844683 0.92 DHPS (0.54) ALDH1A1DHPSHTTEDNRAEDNRB
SCHEMBL7830607 0.90 EDNRA (0.55) ALDH1A1KMT2AMAPTGAAMEN1
SCHEMBL7830604 0.90 EDNRA (0.55) ALDH1A1KMT2AMAPTGAAMEN1
SCHEMBL7839629 0.90 EDNRA (0.50) ALDH1A1DHPSHTTEDNRAEDNRB
SCHEMBL7839633 0.90 EDNRA (0.50) ALDH1A1DHPSHTTEDNRAEDNRB
SCHEMBL7840413 0.88 ALDH1A1 (0.45) ALDH1A1DHPSHTTEDNRAEDNRB
SCHEMBL7840415 0.88 ALDH1A1 (0.45) ALDH1A1DHPSHTTEDNRAEDNRB
SCHEMBL7840232 0.86 ALDH1A1 (0.47) ALDH1A1DHPSHTTEDNRAEDNRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0882719-B1 ARYLETHENESULFONAMIDE DERIVATIVES AND DRUG COMPOSITION CONTAINING THE SAME YAMANOUCHI PHARMA CO LTD (JP) 2001-05-16 EP disclosed
US-6083955-A HAVING A HIGH AFFINITY FOR DRUGS, ESPECIALLY ENDOSERINE RECEPTORS YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 2000-07-04 US disclosed
EP-0882719-A1 ARYLETHENESULFONAMIDE DERIVATIVES AND DRUG COMPOSITION CONTAINING THE SAME YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1998-12-09 EP disclosed