SCHEMBL7843891

SCHEMBL7843891

CCc1ccc(-c2cc(OC)ccn2)cc1N=C(N)N(C(=O)OC(C)(C)C)C(=O)OC(C)(C)C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLAU P00749 2/20 0.37
CCR1 P32246 1/20 0.35
CCR5 P51681 1/20 0.35
CCR8 P51685 1/20 0.35
ALDH1A1 P00352 2/20 0.32
USP2 O75604 2/20 0.32
CYP1A2 P05177 2/20 0.32
CYP3A4 P08684 2/20 0.32
CYP2C19 P33261 2/20 0.32
TSHR P16473 1/20 0.32
ABL1 P00519 1/20 0.31
BCR P11274 1/20 0.31
MAPT P10636 1/20 0.31
HTT P42858 1/20 0.31
RIOK2 Q9BVS4 1/20 0.31
BTK Q06187 1/20 0.30
FAAH O00519 1/20 0.30
CES1 P23141 1/20 0.30
KDM1A O60341 2/20 0.30
HDAC1 Q13547 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7843889 1.00 PLAU (0.37) PLAUCCR1CCR5CCR8ALDH1A1
SCHEMBL7847263 0.82 KDM4E (0.40) PLAUCCR1CCR5CCR8ALDH1A1
SCHEMBL7847265 0.82 KDM4E (0.40) PLAUCCR1CCR5CCR8ALDH1A1
SCHEMBL7842808 0.79 AAK1 (0.37) ABL1BCRMAPTHDAC1
SCHEMBL7843894 0.72 CTSL (0.34) CCR1CCR5CCR8ALDH1A1USP2
SCHEMBL7846734 0.69 CNR1 (0.39) PLAUCCR1CCR5CCR8ABL1
SCHEMBL7230744 0.69 AAK1 (0.40) CCR1CCR5CCR8ABL1BCR
SCHEMBL7846731 0.69 CNR1 (0.39) PLAUCCR1CCR5CCR8ABL1
SCHEMBL7239061 0.69 AAK1 (0.41) PLAUCCR1CCR5CCR8
SCHEMBL7232327 0.69 CCR1 (0.38) PLAUCCR1CCR5CCR8ABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1157022-A1 PYRIDINE COMPOUNDS AND THEIR PHARMACEUTICAL USE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-11-28 EP disclosed
WO-2000049015-A1 PYRIDINE COMPOUNDS AND THEIR PHARMACEUTICAL USE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-08-24 WO disclosed