SCHEMBL7847263

SCHEMBL7847263

COc1ccnc(-c2cccc(/N=C(\N)N(C(=O)OC(C)(C)C)C(=O)OC(C)(C)C)c2)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 2/20 0.40
MAPT P10636 2/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
TP53 P04637 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
PLAU P00749 2/20 0.39
HTR3E A5X5Y0 1/20 0.38
HTR3B O95264 1/20 0.38
HTR3A P46098 1/20 0.38
HTR3D Q70Z44 1/20 0.38
HTR3C Q8WXA8 1/20 0.38
LMNA P02545 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
TAAR1 Q96RJ0 1/20 0.38
CCR1 P32246 1/20 0.37
CCR5 P51681 1/20 0.37
CCR8 P51685 1/20 0.37
WNK1 Q9H4A3 1/20 0.36
LHCGR P22888 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7847265 1.00 KDM4E (0.40) KDM4EALDH1A1MAPTL3MBTL1TP53
SCHEMBL7846734 0.88 CNR1 (0.39) PLAUHTR3EHTR3BHTR3AHTR3D
SCHEMBL7846731 0.88 CNR1 (0.39) PLAUHTR3EHTR3BHTR3AHTR3D
SCHEMBL17560326 0.84 HTR3E (0.55) MAPTL3MBTL1SMN1; SMN2HTR3EHTR3B
SCHEMBL7228914 0.82 SIGMAR1 (0.41) KDM4EALDH1A1MAPTL3MBTL1TP53
SCHEMBL7843889 0.82 PLAU (0.37) KDM4EALDH1A1MAPTPLAULMNA
SCHEMBL7843891 0.82 PLAU (0.37) KDM4EALDH1A1MAPTPLAULMNA
SCHEMBL7229573 0.81 CCR1 (0.40) KDM4EALDH1A1MAPTL3MBTL1TP53
Hydrochloric Acid SCHEMBL7229297 0.78 TAAR1 (0.62) KDM4EALDH1A1MAPTL3MBTL1TP53
SCHEMBL7842304 0.78 TRPV1 (0.37) LHCGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1157022-A1 PYRIDINE COMPOUNDS AND THEIR PHARMACEUTICAL USE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-11-28 EP disclosed
WO-2000049015-A1 PYRIDINE COMPOUNDS AND THEIR PHARMACEUTICAL USE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-08-24 WO disclosed