SCHEMBL7843956

SCHEMBL7843956

Cc1ccnc(-c2ccc(C)c(NC(=NC(=O)OC(C)(C)C)NC(=O)OC(C)(C)C)c2)c1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 11/20 0.39
TP53 P04637 1/20 0.38
MAPT P10636 1/20 0.38
THRB P10828 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
LMNA P02545 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
CYP1A2 P05177 1/20 0.37
POLB P06746 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C19 P33261 1/20 0.37
ALDH1A1 P00352 1/20 0.37
CNR1 P21554 1/20 0.36
BRD9 Q9H8M2 1/20 0.36
ACACB O00763 1/20 0.36
ACACA Q13085 1/20 0.36
MAPK14 Q16539 1/20 0.36
SMO Q99835 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7853175 0.89 KDM4E (0.40) AAK1TP53MAPTTHRBTDP1
SCHEMBL7841629 0.85 ACACB (0.35) AAK1CNR1ACACBACACA
SCHEMBL7846551 0.84 CNR1 (0.52) TP53MAPTTDP1LMNANPSR1
SCHEMBL7238064 0.81 AAK1 (0.41) AAK1CNR1ACACBACACA
SCHEMBL7845048 0.79 KDR (0.41)
SCHEMBL7846741 0.79 AAK1 (0.38) AAK1TP53THRBCYP1A2CYP3A4
SCHEMBL23246323 0.78 L3MBTL1 (0.44) MAPTLMNANPSR1POLBALDH1A1
SCHEMBL29707255 0.78 L3MBTL1 (0.44) MAPTLMNANPSR1POLBALDH1A1
SCHEMBL28739389 0.78 ALDH1A1 (0.44) MAPTTDP1LMNAALDH1A1
SCHEMBL23246313 0.78 L3MBTL1 (0.44) MAPTLMNANPSR1POLBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1157022-A1 PYRIDINE COMPOUNDS AND THEIR PHARMACEUTICAL USE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-11-28 EP disclosed
WO-2000049015-A1 PYRIDINE COMPOUNDS AND THEIR PHARMACEUTICAL USE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-08-24 WO disclosed