SCHEMBL7844289

SCHEMBL7844289

COc1ccnc(-c2ccc(C3OCCO3)c(NC(=NC(=O)OC(C)(C)C)NC(=O)OC(C)(C)C)c2)c1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACACB O00763 1/20 0.34
ACACA Q13085 1/20 0.34
AAK1 Q2M2I8 7/20 0.33
CHRM1 P11229 1/20 0.32
BTK Q06187 1/20 0.32
ABL1 P00519 1/20 0.31
BCR P11274 1/20 0.31
BACE1 P56817 1/20 0.31
KCNH2 Q12809 1/20 0.31
USP30 Q70CQ3 1/20 0.31
DYRK1A Q13627 1/20 0.31
ATR Q13535 1/20 0.31
CCR1 P32246 1/20 0.31
CCR5 P51681 1/20 0.31
CCR8 P51685 1/20 0.31
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30
GLA P06280 1/20 0.30
GAA P10253 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7841629 0.90 ACACB (0.35) ACACBACACAAAK1
SCHEMBL7853175 0.84 KDM4E (0.40) AAK1DYRK1ACCR1CCR5CCR8
SCHEMBL7238123 0.84 ABL1 (0.35) ACACBACACAAAK1CHRM1BTK
SCHEMBL7846741 0.84 AAK1 (0.38) AAK1ATRCCR1CCR5CCR8
SCHEMBL7845048 0.84 KDR (0.41)
SCHEMBL7843005 0.80 CYP17A1 (0.41)
SCHEMBL7833912 0.78 CNR1 (0.34) ACACBACACAAAK1ABL1BCR
SCHEMBL7240473 0.75 CCR1 (0.33) AAK1BTKDYRK1AATRCCR1
SCHEMBL7843956 0.74 AAK1 (0.39) ACACBACACAAAK1ALDH1A1LMNA
SCHEMBL7231706 0.74 AAK1 (0.36) ACACBACACAAAK1ABL1BCR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1157022-A1 PYRIDINE COMPOUNDS AND THEIR PHARMACEUTICAL USE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-11-28 EP disclosed
WO-2000049015-A1 PYRIDINE COMPOUNDS AND THEIR PHARMACEUTICAL USE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-08-24 WO disclosed