SCHEMBL7845162

SCHEMBL7845162

O=C(c1c[nH]c2ccc(C#CCO)cc2c1=O)N(Cc1ccc(Cl)cc1)C1CC1

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 4/20 0.39
GABRB2 P47870 4/20 0.39
CFTR P13569 1/20 0.37
HAT1 O14929 1/20 0.37
EP300 Q09472 1/20 0.37
AGER Q15109 1/20 0.37
C5AR1 P21730 1/20 0.36
POLB P06746 1/20 0.36
NSD2 O96028 1/20 0.36
ALDH1A1 P00352 1/20 0.35
NHERF1 O14745 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7843694 0.85 GAA (0.46) GABRA1GABRB2CFTRPOLBALDH1A1
SCHEMBL6670139 0.84 CFTR (0.39) GABRA1GABRB2CFTRPOLBNHERF1
SCHEMBL7845927 0.84 HAT1 (0.44) GABRA1GABRB2CFTRHAT1EP300
SCHEMBL7833923 0.84 CFTR (0.45) GABRA1GABRB2CFTRPOLBALDH1A1
SCHEMBL7843172 0.83 GABRA1 (0.40) GABRA1GABRB2CFTRALDH1A1
SCHEMBL7860741 0.83 GABRA1 (0.39) GABRA1GABRB2CFTRPOLB
SCHEMBL7847436 0.81 KDM4E (0.44) GABRA1GABRB2CFTRPOLBALDH1A1
SCHEMBL7842246 0.81 KDM4E (0.44) GABRA1GABRB2CFTRPOLBALDH1A1
SCHEMBL7835904 0.81 GABRA1 (0.40) GABRA1GABRB2
SCHEMBL7845109 0.80 CFTR (0.42) GABRA1GABRB2CFTRPOLBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140850-A1 QUINOLINECARBOXAMIDES AS ANTIVIRAL AGENTS PHARMACIA & UPJOHN COMPANY (US) 2001-10-10 EP disclosed
WO-2000040561-A1 QUINOLINECARBOXAMIDES AS ANTIVIRAL AGENTS PHARMACIA & UPJOHN COMPANY (US) 2000-07-13 WO disclosed