SCHEMBL7845462

SCHEMBL7845462

S=C1C=NSc2ccccc2C1

nearest known ligand 0.34

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.34
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34
MEN1 O00255 1/20 0.31
NPC1 O15118 1/20 0.31
HSP90AA1 P07900 1/20 0.31
MAPT P10636 1/20 0.31
THRB P10828 1/20 0.31
HK1 P19367 1/20 0.31
MAPK1 P28482 1/20 0.31
RECQL P46063 1/20 0.31
RAB9A P51151 1/20 0.31
GALK1 P51570 1/20 0.31
BLM P54132 1/20 0.31
KMT2A Q03164 1/20 0.31
HKDC1 Q2TB90 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL720559 0.81 ALDH1A1 (0.42) KDM4EALDH1A1HPGDMEN1MAPT
Hydrochloric Acid SCHEMBL3154489 0.79 ALDH1A1 (0.41) KDM4EALDH1A1HPGDMEN1MAPT
SCHEMBL7837771 0.77 KDM4E (0.34) KDM4EALDH1A1HPGD
SCHEMBL1868060 0.68 ALDH1A1 (0.36) KDM4EALDH1A1HPGDMEN1MAPT
SCHEMBL3081411 0.67 ALDH1A1 (0.38) KDM4EALDH1A1HPGDMEN1MAPT
SCHEMBL8275 0.67 RYR2 (0.31) KDM4EALDH1A1HPGD
Hydrochloric Acid SCHEMBL6424274 0.65 RYR2 (0.31)
SCHEMBL7730853 0.65 TRPA1 (0.59) KDM4EHPGDMEN1NPC1HSP90AA1
SCHEMBL7994953 0.65 ALDH1A1 (0.46) KDM4EALDH1A1HPGDMEN1MAPT
Thioxanthene SCHEMBL27774542 0.65 ALDH1A1 (0.59) KDM4EALDH1A1HPGDMEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1155007-A2 1,2-BENZOTHIAZEPINES FOR THE TREATMENT OF HYPERLIPIDEMIC DISEASES G.D. Searle LLC (US) 2001-11-21 EP disclosed
WO-2000047568-A2 1,2-BENZOTHIAZEPINES FOR THE TREATMENT OF HYPERLIPIDEMIC DISEASES G.D. SEARLE LLC (US) 2000-08-17 WO disclosed