SCHEMBL7845819

SCHEMBL7845819

CCOCCn1cc(C(=O)CN2CCC(n3c(C)nc4cnccc43)CC2)c2c(OC(=O)OC)cccc21

nearest known ligand 0.79

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 4/20 0.44
CYP2D6 P10635 1/20 0.44
MAPK1 P28482 2/20 0.39
UBE2N P61088 2/20 0.39
NPSR1 Q6W5P4 2/20 0.39
GLA P06280 1/20 0.39
HSD17B10 Q99714 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
KDR P35968 1/20 0.38
ALDH1A1 P00352 1/20 0.37
CYP3A4 P08684 1/20 0.37
USP2 O75604 1/20 0.36
MCHR1 Q99705 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7835350 0.90 CYP2D6 (0.44) CCR5CYP2D6
SCHEMBL7835611 0.90 CCR5 (0.46) CCR5CYP2D6MAPK1UBE2NNPSR1
SCHEMBL7834134 0.88 CCR5 (0.45) CCR5CYP2D6MAPK1UBE2NNPSR1
SCHEMBL7846720 0.81 CCR5 (0.46) CCR5CYP2D6MAPK1UBE2NNPSR1
SCHEMBL9056669 0.74 CCR5 (0.38) CCR5CYP2D6CYP3A4
SCHEMBL7848279 0.72 CYP2D6 (0.47) CCR5CYP2D6
SCHEMBL7845147 0.71 CCR5 (0.45) CCR5CYP2D6MAPK1UBE2NNPSR1
SCHEMBL7834484 0.71
SCHEMBL7834120 0.71 CYP2D6 (0.46) CCR5CYP2D6MAPK1UBE2NNPSR1
SCHEMBL7841961 0.70 CCR5 (0.43) CCR5CYP2D6MAPK1UBE2NNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0821685-B1 INDOLE-3-CARBONYL AND INDOLE-3-SULFONYL DERIVATIVES AS PLATELET ACTIVATING FACTOR ANTAGONISTS ABBOTT LAB (US) 2001-10-04 EP claimed